SCHEMBL7725428

SCHEMBL7725428

COc1ccc(CCN)c(C)c1OCC1CC1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.41
ADRA1A P35348 1/20 0.41
HTR2A P28223 3/20 0.39
PDE4B Q07343 2/20 0.39
PDE4D Q08499 1/20 0.38
HTR7 P34969 1/20 0.38
HTR6 P50406 1/20 0.38
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303296 0.80 TAAR1 (0.52) TAAR1ADRA1AHTR2ACYP1A2
SCHEMBL4384909 0.77 TAAR1 (0.55) TAAR1ADRA1AALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL1437384 0.75 TAAR1 (0.53) TAAR1ADRA1AALDH1A1CYP1A2
SCHEMBL20970869 0.74 HTR2A (0.64) TAAR1HTR2APDE4BHTR7HTR6
SCHEMBL2587027 0.72 SMN1; SMN2 (0.57) PDE4BPDE4DALDH1A1CYP1A2
SCHEMBL34463016 0.71 TAAR1 (0.52) TAAR1ADRA1AHTR2ACYP1A2
SCHEMBL1253168 0.70 AOC3 (0.64) TAAR1ADRA1AHTR2AALDH1A1CYP1A2
SCHEMBL16011771 0.69 SMN1; SMN2 (0.44) HTR2APDE4BPDE4DHTR7HTR6
SCHEMBL2581701 0.69 PDE4D (0.47) ADRA1AHTR2APDE4BPDE4DHTR7
Hydrochloric Acid SCHEMBL7366474 0.69 AOC3 (0.62) TAAR1ADRA1AHTR2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403805-B1 SUCH AS 1-((1-(3-(CYCLOPENTYLOXY)-4-METHOXYPHENYL) CYCLOPROPYL)METHYL)-1,3-DIHYDRO-2H-IMIDAZOL-2-ONE FOR ALLERGIES, ATOPIC AND INFLAMMATORY DISEASES WHEREIN ACTIVITY OF PHOSPHODIESTERASE IS ALTERED JANSSEN PHARMACEUTICA N.V. (BE) 2002-06-11 US disclosed