SCHEMBL7732374

SCHEMBL7732374

CCCCCCCCCCC1CCN(CCCOc2ccc(-c3ccc(C(C)=O)cc3)cc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 6/20 0.58
HRH1 P35367 6/20 0.58
HRH3 Q9Y5N1 11/20 0.56
KDM4E B2RXH2 1/20 0.56
KCNH2 Q12809 1/20 0.52
THRA P10827 1/20 0.51
THRB P10828 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7739073 1.00 HRH2 (0.58) HRH2HRH1HRH3KDM4EKCNH2
SCHEMBL7732361 1.00 HRH2 (0.58) HRH2HRH1HRH3KDM4EKCNH2
SCHEMBL7738905 0.94 HRH2 (0.55) HRH2HRH1HRH3KDM4ETHRA
SCHEMBL7741808 0.87 HRH2 (0.57) HRH2HRH1HRH3KDM4EKCNH2
SCHEMBL13472015 0.80 HRH2 (0.56) HRH2HRH1HRH3KCNH2THRA
SCHEMBL491570 0.79 HRH3 (0.72) HRH2HRH1HRH3KDM4E
SCHEMBL15177348 0.79 GAA (0.77) THRATHRB
SCHEMBL12243177 0.79 GAA (0.77) THRATHRB
SCHEMBL9000300 0.79 GAA (0.77) THRATHRB
SCHEMBL7739031 0.79 GAA (0.77) THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7790744-B2 Cyclic peptide antifungal agents and process for preparation thereof ELI LILLY AND COMPANY (US) 2010-09-07 US disclosed
US-7790744-B2 Cyclic peptide antifungal agents and process for preparation thereof ELI LILLY AND COMPANY (US) 2010-09-07 US disclosed
US-6743777-B1 TRISPHENYL ACYL DERIVATIVES OF THE ECHINOCANDIN CLASS; CANDIDA ALBICANS; ANTIFUNGAL AND ANTIPARASITIC; CYCLIC HEXAPEPTIDES HAVING UNIQUE SIDE CHAIN ACYL GROUP ELI LILLY AND COMPANY 2004-06-01 US disclosed
US-6743777-B1 TRISPHENYL ACYL DERIVATIVES OF THE ECHINOCANDIN CLASS; CANDIDA ALBICANS; ANTIFUNGAL AND ANTIPARASITIC; CYCLIC HEXAPEPTIDES HAVING UNIQUE SIDE CHAIN ACYL GROUP ELI LILLY AND COMPANY 2004-06-01 US disclosed