SCHEMBL7735787

SCHEMBL7735787

C[SiH](C)O[C@](C)(CCC(C)(C)C)n1cnc(-c2cccnc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 6/20 0.48
CYP2C19 P33261 4/20 0.48
CYP3A4 P08684 4/20 0.48
CYP2E1 P05181 3/20 0.48
CYP2C9 P11712 3/20 0.48
CYP2B6 P20813 3/20 0.48
CYP2D6 P10635 2/20 0.42
HSP90AA1 P07900 4/20 0.40
HSP90AB1 P08238 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CYP19A1 P11511 2/20 0.34
CYP1A2 P05177 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
P4HTM Q9NXG6 1/20 0.34
FYN P06241 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15471025 0.73 CYP2A6 (0.69) CYP2A6CYP2C19CYP3A4CYP2E1CYP2C9
SCHEMBL4869247 0.72 CYP2A6 (0.59) CYP2A6CYP2C19CYP3A4CYP2E1CYP2C9
SCHEMBL5507651 0.72 CYP2A6 (0.56) CYP2A6CYP2C19CYP3A4CYP2E1CYP2C9
SCHEMBL4864745 0.71 CYP2A6 (0.52) CYP2A6CYP2C19CYP3A4CYP2E1CYP2C9
SCHEMBL4870330 0.71 CYP2A6 (0.52) CYP2A6CYP2C19CYP3A4CYP2E1CYP2C9
SCHEMBL4862008 0.71 CYP2A6 (0.54) CYP2A6CYP2C19CYP3A4CYP2E1CYP2C9
SCHEMBL4870983 0.70 CYP2A6 (0.48) CYP2A6CYP2C19CYP3A4CYP2E1CYP2C9
SCHEMBL13527034 0.70 CYP2A6 (0.64) CYP2A6CYP2C19CYP3A4CYP2E1CYP2C9
SCHEMBL17688341 0.67 CYP2A6 (0.55) CYP2A6CYP2C19CYP3A4CYP2E1CYP2C9
SCHEMBL24809712 0.67 CYP2A6 (0.49) CYP2A6CYP2C19CYP3A4CYP2E1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403776-B1 TREATING ANTIBIOTIC COMPOUND WITH NUCLEOPHILE TO CLEAVE PROTECTING GROUP FROM HYDROXYL GROUP PFIZER INC. 2002-06-11 US disclosed
EP-1088828-A2 Synthesis of carbamate ketolide antibiotics Pfizer Products Inc. (US) 2001-04-04 EP disclosed