SCHEMBL7737157

SCHEMBL7737157

CCC[C@H]1CC[C@H](CCc2cccc(C(=O)O)c2F)CC1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 8/20 0.41
CYP2C9 P11712 1/20 0.38
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
CLCN2 P51788 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
KAT6A Q92794 1/20 0.36
HMGB1 P09429 1/20 0.36
CXCR5 P32302 1/20 0.36
FOLH1 Q04609 1/20 0.36
NFE2L2 Q16236 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7737160 1.00 MRGPRX4 (0.41) MRGPRX4CYP2C9HTR2AHTR2CCLCN2
SCHEMBL7736471 0.88 HTR2A (0.37) MRGPRX4CYP2C9HTR2AHTR2CALDH1A1
SCHEMBL7736468 0.88 HTR2A (0.37) MRGPRX4CYP2C9HTR2AHTR2CALDH1A1
SCHEMBL9561945 0.88 CYP2C9 (0.39) CYP2C9HTR2AHTR2CALDH1A1LMNA
SCHEMBL9561955 0.88 CYP2C9 (0.39) CYP2C9HTR2AHTR2CALDH1A1LMNA
SCHEMBL8470973 0.86 FOLH1 (0.50) CYP2C9HTR2AHTR2CCLCN2ALDH1A1
SCHEMBL8470980 0.86 FOLH1 (0.50) CYP2C9HTR2AHTR2CCLCN2ALDH1A1
SCHEMBL8447505 0.85 FOLH1 (0.49) CYP2C9HTR2AHTR2CCLCN2ALDH1A1
SCHEMBL8776357 0.83 CXCR5 (0.36) CYP2C9HTR2AHTR2CALDH1A1LMNA
SCHEMBL8776360 0.83 CXCR5 (0.36) CYP2C9HTR2AHTR2CALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6468606-B1 LOW VISCOSITY, HIGH DIELECTRIC ANISOTROPY, LOW OPTICAL ANISOTROPY, EXCELLENT LOW TEMPERATURE COMPATIBILITY WITH OTHER LIQUID CRYSTALLINE COMPOUNDS; 3,4,5-TRIFLUOROPHENYL-(2-FLUORO-4-(TRANS-4-PROPYLCYCLOHEXYL))BENZOATE CHISSO CORPORATION (JP) 2002-10-22 US disclosed
EP-0808825-B1 PHENYL BENZOATE DERIVATIVES AND LIQUID CRYSTAL COMPOSITIONS CHISSO CORP (JP) 2001-09-12 EP disclosed
US-5922243-A LOW VISCOSITY, HIGH DIELECTRIC AND LOW OPTICAL ANISOTROPY, EXCELLENT COMPATIBILITY CHISSO CORPORATION (JP) 1999-07-13 US disclosed
EP-0808825-A1 PHENYL BENZOATE DERIVATIVES AND LIQUID CRYSTAL COMPOSITIONS CHISSO CORPORATION (JP) 1997-11-26 EP disclosed