SCHEMBL7738801

SCHEMBL7738801

CC(=O)c1cc(=O)c2ccccc2[nH]1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.72
HPGD P15428 5/20 0.72
CYP1A2 P05177 3/20 0.72
GAA P10253 2/20 0.72
HSD17B10 Q99714 2/20 0.72
CYP2C19 P33261 2/20 0.72
ALDH1A1 P00352 2/20 0.72
MEN1 O00255 2/20 0.72
MAPK1 P28482 2/20 0.72
KMT2A Q03164 2/20 0.72
GRIN2D O15399 1/20 0.72
GRIN3B O60391 1/20 0.72
GLA P06280 1/20 0.72
AHR P35869 1/20 0.72
CHRNA7 P36544 1/20 0.72
GRIN1 Q05586 1/20 0.72
GRIN2A Q12879 1/20 0.72
GRIN2B Q13224 1/20 0.72
GRIN2C Q14957 1/20 0.72
GRIN3A Q8TCU5 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Transtorine SCHEMBL5144405 0.84 KDM4E (1.00) KDM4EHPGDCYP1A2GAAHSD17B10
Transtorine SCHEMBL29366068 0.84 KDM4E (1.00) KDM4EHPGDCYP1A2GAAHSD17B10
Transtorine SCHEMBL29841751 0.82 KDM4E (0.96) KDM4EHPGDCYP1A2GAAHSD17B10
SCHEMBL3290252 0.82 KDM4E (0.72) KDM4EHPGDCYP1A2GAAHSD17B10
SCHEMBL57291 0.81 KDM4E (0.66) KDM4EHPGDCYP1A2GAAHSD17B10
SCHEMBL31243255 0.81 KDM4E (0.66) KDM4EHPGDCYP1A2GAAHSD17B10
SCHEMBL13545149 0.81 KDM4E (0.66) KDM4EHPGDCYP1A2GAAHSD17B10
SCHEMBL13543209 0.81 HPGD (0.66) KDM4EHPGDCYP1A2GAAHSD17B10
Transtorine SCHEMBL30853453 0.81 KDM4E (0.70) KDM4EHPGDCYP1A2GAAHSD17B10
SCHEMBL31437284 0.78 KDM4E (0.62) KDM4EHPGDCYP1A2GAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7790744-B2 Cyclic peptide antifungal agents and process for preparation thereof ELI LILLY AND COMPANY (US) 2010-09-07 US disclosed
US-6743777-B1 TRISPHENYL ACYL DERIVATIVES OF THE ECHINOCANDIN CLASS; CANDIDA ALBICANS; ANTIFUNGAL AND ANTIPARASITIC; CYCLIC HEXAPEPTIDES HAVING UNIQUE SIDE CHAIN ACYL GROUP ELI LILLY AND COMPANY 2004-06-01 US disclosed