SCHEMBL7745332

SCHEMBL7745332

CC(O)[C@H]1CC[C@H]2[C@@H]3CCC4NC(=O)CC[C@]4(C)[C@H]3CC[C@]12C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 4/20 0.69
SRD5A1 P18405 3/20 0.69
AR P10275 1/20 0.54
CYP17A1 P05093 2/20 0.53
KDM4E B2RXH2 1/20 0.53
MAPT P10636 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7745329 1.00 SRD5A2 (0.69) SRD5A2SRD5A1ARCYP17A1KDM4E
SCHEMBL8074664 0.88 SRD5A2 (0.69) SRD5A2SRD5A1AR
SCHEMBL8074665 0.88 SRD5A2 (0.69) SRD5A2SRD5A1AR
SCHEMBL8063981 0.85 SRD5A2 (0.75) SRD5A2SRD5A1
SCHEMBL8063986 0.85 SRD5A2 (0.75) SRD5A2SRD5A1
SCHEMBL7382153 0.82 SRD5A2 (0.71) SRD5A2SRD5A1CYP17A1KDM4EMAPT
SCHEMBL7382151 0.82 SRD5A2 (0.71) SRD5A2SRD5A1CYP17A1KDM4EMAPT
SCHEMBL4269548 0.82 SRD5A2 (0.64) SRD5A2SRD5A1AR
SCHEMBL4269554 0.82 SRD5A2 (0.64) SRD5A2SRD5A1AR
SCHEMBL5682764 0.82 SRD5A2 (0.64) SRD5A2SRD5A1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0649306-B1 ESTER DERIVATIVES OF 4-AZA-STEROIDS MERCK & CO INC (US) 2001-01-10 EP disclosed
US-5693809-A PREGNANES FOR TREATING ALOPECIA, ACNE AND SKIN DISORDER MERCK & CO., INC. (US) 1997-12-02 US disclosed
US-5610162-A ENZYME INHIBITORS MERCK & CO., INC. (US) 1997-03-11 US disclosed
EP-0649306-A4 ESTER DERIVATIVES OF 4-AZA-STEROIDS. MERCK & CO INC (US) 1995-08-23 EP disclosed
EP-0649306-A1 ESTER DERIVATIVES OF 4-AZA-STEROIDS MERCK & CO. INC. (US) 1995-04-26 EP disclosed
WO-1993023041-A1 ESTER DERIVATIVES OF 4-AZA-STEROIDS MERCK & CO., INC. (US) 1993-11-25 WO disclosed
WO-1993023039-A1 SUBSTITUTED 4-AZA-5A-ANDROSTAN-ONES AS 5A-REDUCTASE INHIBITORS MERCK & CO., INC. (US) 1993-11-25 WO disclosed