SCHEMBL7745840

SCHEMBL7745840

COc1ccc2c(c1C)/C(=C/c1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1)C(=O)N2

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 5/20 0.57
EGFR P00533 3/20 0.57
IGF1R P08069 1/20 0.57
DHFR P00374 1/20 0.48
CTRC Q99895 1/20 0.47
EEF2K O00418 1/20 0.46
SRC P12931 1/20 0.46
GAA P10253 1/20 0.45
PLK4 O00444 1/20 0.44
PLK1 P53350 1/20 0.44
RET P07949 1/20 0.44
PTGS2 P35354 4/20 0.44
PTGS1 P23219 3/20 0.44
LRRK2 Q5S007 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5364049 0.84 ERBB2 (0.59) ERBB2EGFRIGF1RCTRCEEF2K
SCHEMBL5366009 0.81 ERBB2 (0.62) ERBB2EGFRIGF1RPLK4PLK1
SCHEMBL5360968 0.80 EGFR (0.54) ERBB2EGFRIGF1RCTRCEEF2K
SCHEMBL7317553 0.79 ERBB2 (0.68) ERBB2EGFRIGF1RCTRCEEF2K
SCHEMBL7317561 0.79 ERBB2 (0.68) ERBB2EGFRIGF1RCTRCEEF2K
SCHEMBL5367617 0.79 ERBB2 (0.53) ERBB2EGFRIGF1RCTRCEEF2K
SCHEMBL5366011 0.78 ERBB2 (0.61) ERBB2EGFRIGF1RPLK4PLK1
SCHEMBL5362776 0.76 ERBB2 (0.67) ERBB2EGFRIGF1RPLK4PLK1
SCHEMBL7311443 0.76 EGFR (0.67) ERBB2EGFRIGF1RCTRCEEF2K
SCHEMBL7311437 0.76 EGFR (0.67) ERBB2EGFRIGF1RCTRCEEF2K

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001021166-A1 TREATMENT AND PREVENTION OF HEPATIC DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2001-03-29 WO disclosed