Broussonin A

Broussonin A

SCHEMBL774802

COc1ccc(CCCc2ccc(O)cc2)c(O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 1.00
CYP19A1 P11511 1/20 1.00
ESR2 Q92731 1/20 1.00
CALM1 P0DP23 3/20 0.72
POLB P06746 1/20 0.56
IGF1R P08069 1/20 0.55
ALOX15 P16050 1/20 0.55
SLC28A3 Q9HAS3 1/20 0.49
TYR P14679 1/20 0.49
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736569 0.90 ESR1 (0.82) ESR1CYP19A1ESR2CALM1POLB
SCHEMBL13084317 0.88 ESR1 (0.78) ESR1CYP19A1ESR2CALM1POLB
SCHEMBL9202466 0.88 ESR1 (0.78) ESR1CYP19A1ESR2CALM1IGF1R
Broussonin E SCHEMBL31510414 0.85 CYP19A1 (0.74) ESR1CYP19A1ESR2CALM1POLB
Broussonin E SCHEMBL6825353 0.85 CYP19A1 (0.74) ESR1CYP19A1ESR2CALM1POLB
SCHEMBL227115 0.85 ESR1 (0.73) ESR1CYP19A1ESR2CALM1POLB
SCHEMBL6822966 0.83 ESR1 (0.70) ESR1CYP19A1ESR2IGF1RALOX15
SCHEMBL30576426 0.83 ESR1 (0.70) ESR1CYP19A1ESR2CALM1POLB
SCHEMBL1850095 0.83 ESR1 (0.70) ESR1CYP19A1ESR2CALM1POLB
SCHEMBL25328659 0.82 ESR1 (0.69) ESR1CYP19A1ESR2CALM1IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250195452-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE IATERION, INC. 2025-06-19 US claimed
EP-4561582-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE Iaterion, Inc. (US) 2025-06-04 EP claimed
WO-2024026037-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE IATERION, INC. (US) 2024-02-01 WO claimed
WO-2010120029-A1 COMPOSITION COMPRISING THE EXTRACT OF ANEMARRHENA ASPHODELOIDES BUNGE OR THE COMPOUNDS ISOLATED FROM THE SAME FOR PREVENTING AND TREATING LIPID METABOLISM DISORDER EWHA UNIVERSITY - INDUSTRY COLLABORATION FOUNDATION (KR) 2010-10-21 WO claimed
US-6737439-B2 ACTIVE CANCER CHEMOPREVENTATIVE AND TREATING AGENTS IN MAMMALS, INCLUDING HUMANS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2004-05-18 US claimed
US-20030125377-A1 Aromatase inhibitors from Broussonetia papyrifera BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS THE 2003-07-03 US claimed
WO-2003013554-A2 AROMATASE INHIBITORS FROM BROUSSONETIA PAPYRIFERA THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2003-02-20 WO claimed
US-20250195452-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE IATERION, INC. 2025-06-19 US disclosed
EP-4561582-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE Iaterion, Inc. (US) 2025-06-04 EP disclosed
CN-119604294-A ERbeta estrogenic compounds and methods of use 益特瑞恩公司 2025-03-11 CN disclosed
WO-2024026037-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE IATERION, INC. (US) 2024-02-01 WO disclosed
US-11857657-B2 Diarylalkanes as potent inhibitors of binuclear enzymes UNIGEN, INC. (US) 2024-01-02 US disclosed
CN-109134205-B Diarylalkanes as potent inhibitors of binuclear enzymes 尤尼根公司 2022-07-19 CN disclosed
CN-1993114-A Diarylalkanes as potent inhibitors of binuclear enzymes UNIGEN PHARMACEUTICALS INC (US) 2007-07-04 CN disclosed
EP-1748767-A1 DIARYLALKANES AS POTENT INHIBITORS OF BINUCLEAR ENZYMES Unigen Pharmaceuticals, Inc. (US) 2007-02-07 EP disclosed
WO-2005117849-A1 DIARYLALKANES AS POTENT INHIBITORS OF BINUCLEAR ENZYMES UNIGEN PHARMACEUTICALS, INC. (US) 2005-12-15 WO disclosed
US-20050267047-A1 Diarylalkanes as potent inhibitors of binuclear enzymes UNIGEN PHARMACEUTICALS, INC. (US) 2005-12-01 US disclosed
US-6737439-B2 ACTIVE CANCER CHEMOPREVENTATIVE AND TREATING AGENTS IN MAMMALS, INCLUDING HUMANS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2004-05-18 US disclosed
US-20030125377-A1 Aromatase inhibitors from Broussonetia papyrifera BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS THE 2003-07-03 US disclosed
WO-2003013554-A2 AROMATASE INHIBITORS FROM BROUSSONETIA PAPYRIFERA THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2003-02-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030125377-A1 Aromatase inhibitors from Broussonetia papyrifera CYP19A1, HSD17B11, CYP17A1 ESR1 44/4885CYP19A1 1/4885ESR2 75/4885
US-20050267047-A1 Diarylalkanes as potent inhibitors of binuclear enzymes TYR, DDT, HAAO ESR1 3513/4885CYP19A1 203/4885ESR2 3995/4885
US-20250195452-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE ESR2, ESR1, ESRRB ESR1 2/4885CYP19A1 9/4885ESR2 1/4885
US-11857657-B2 Diarylalkanes as potent inhibitors of binuclear enzymes TYR, DDT, HAAO ESR1 3513/4885CYP19A1 203/4885ESR2 3995/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.