SCHEMBL7753475

SCHEMBL7753475

Nc1nc(Nc2ccccc2)sc1-c1cc(F)c(C=O)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 9/20 0.46
CCNA2 P20248 8/20 0.46
MAPT P10636 8/20 0.44
CDK5 Q00535 5/20 0.44
CDK5R1 Q15078 5/20 0.44
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
GSK3B P49841 3/20 0.44
GSK3A P49840 1/20 0.44
MAPK14 Q16539 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
LMNA P02545 4/20 0.44
PSMD14 O00487 1/20 0.44
TP53 P04637 2/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7753473 0.82 CDK2 (0.45) CDK2CCNA2MAPTCDK5CDK5R1
SCHEMBL1248421 0.76 CCNA2 (0.49) CDK2CCNA2MAPTCDK5CDK5R1
SCHEMBL1250520 0.75 MAPT (0.45) CDK2CCNA2MAPTCDK5CDK5R1
SCHEMBL7756995 0.73 MAPT (0.68) CDK2CCNA2MAPTCDK5CDK5R1
SCHEMBL1250757 0.72 MAPT (0.52) CDK2CCNA2MAPTCDK5CDK5R1
SCHEMBL1249747 0.72 MAPT (0.46) CDK2CCNA2MAPTCDK5CDK5R1
SCHEMBL27609556 0.72 CCNA2 (0.59) CDK2CCNA2MAPTCDK5CDK5R1
SCHEMBL1248135 0.72 MAPT (0.45) CDK2CCNA2MAPTCDK5CDK5R1
SCHEMBL1248186 0.71 MAPT (0.45) CDK2CCNA2MAPTCDK5CDK5R1
SCHEMBL1250063 0.71 MAPT (0.44) CDK2CCNA2MAPTCDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001056567-A1 2,4-DIAMINOTHIAZOLE DERIVATIVES AND THEIR USE AS GLYCOGEN SYNTHASE KINASE-3 (GSK-3) INHIBITORS NOVO NORDISK A/S (DK) 2001-08-09 WO disclosed