SCHEMBL7758348

SCHEMBL7758348

CC(=O)n1ccc2cc(C(=O)NC(C)(C)C)ccc21

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.49
POLB P06746 1/20 0.49
NOTUM Q6P988 1/20 0.47
CYP11B1 P15538 3/20 0.44
CYP11B2 P19099 3/20 0.44
CACNA1B Q00975 1/20 0.44
PPARG P37231 2/20 0.43
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MAOB P27338 1/20 0.40
LMNA P02545 2/20 0.39
KMT2A Q03164 1/20 0.39
IMPDH2 P12268 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6827828 0.81 IDH1 (0.47) MAPTPOLBALDH1A1TP53LMNA
SCHEMBL5066779 0.79 NOTUM (0.56) NOTUMCYP11B1CYP11B2PPARGALDH1A1
SCHEMBL7758376 0.77 NOTUM (0.59) NOTUMCYP11B1CYP11B2PPARGALDH1A1
SCHEMBL10837082 0.72 NOTUM (0.59) MAPTNOTUMCYP11B1CYP11B2ALDH1A1
SCHEMBL20812513 0.71 MAPT (0.59) MAPTPOLBCACNA1BALDH1A1HPGD
SCHEMBL28189196 0.71 NOTUM (0.54) NOTUMCYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL12749675 0.70 NOTUM (0.58) NOTUMCYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL7759631 0.70 NPC1 (0.55) ALDH1A1KDM4ETP53LMNAKMT2A
SCHEMBL853076 0.70 NOTUM (0.58) NOTUMCYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL31607288 0.70 NOTUM (0.58) NOTUMCYP11B1CYP11B2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077699-A1 AMIDE THERAPEUTICS FOR THE TREATMENT OF INFLAMMATORY BOWEL DISEASE CENTAUR PHARMACEUTICALS, INC. (US) 2001-02-28 EP claimed
WO-1999059582-A1 AMIDE THERAPEUTICS FOR THE TREATMENT OF INFLAMMATORY BOWEL DISEASE CENTAUR PHARMACEUTICALS, INC. (US) 1999-11-25 WO claimed
US-6271265-B1 N-TERT-BUTYL-2-HYDROXYBENZAMIDE FOR INFLAMMATORY BOWEL DISEASE CENTAUR PHARMACEUTICALS, INC. 2001-08-07 US disclosed
EP-1077699-A1 AMIDE THERAPEUTICS FOR THE TREATMENT OF INFLAMMATORY BOWEL DISEASE CENTAUR PHARMACEUTICALS, INC. (US) 2001-02-28 EP disclosed
WO-1999059582-A1 AMIDE THERAPEUTICS FOR THE TREATMENT OF INFLAMMATORY BOWEL DISEASE CENTAUR PHARMACEUTICALS, INC. (US) 1999-11-25 WO disclosed