SCHEMBL7767367

SCHEMBL7767367

CCOC(=O)c1ccc2[nH]c(=O)sc2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.65
ALDH1A1 P00352 6/20 0.58
KDM4E B2RXH2 4/20 0.58
HSD17B10 Q99714 4/20 0.58
HPGD P15428 3/20 0.58
MAPK1 P28482 2/20 0.58
POLB P06746 1/20 0.58
MAPT P10636 5/20 0.56
RAB9A P51151 4/20 0.56
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
LMNA P02545 2/20 0.52
HTT P42858 1/20 0.52
CA12 O43570 2/20 0.51
CA1 P00915 2/20 0.51
CA2 P00918 2/20 0.51
CA7 P43166 2/20 0.51
CA9 Q16790 2/20 0.51
CA14 Q9ULX7 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28097716 0.84 PDE3B (0.57) HCRTR1ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL13302168 0.84 HCRTR1 (0.59) HCRTR1ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL8781331 0.84 HCRTR1 (0.59) HCRTR1ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL11537592 0.83 HCRTR1 (0.56) HCRTR1ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL9483042 0.81 ESR1 (0.52) HCRTR1MAPTSMN1; SMN2LMNAHTT
SCHEMBL20746469 0.80 HCRTR1 (0.56) HCRTR1ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL9484788 0.80 ESR1 (0.48) HCRTR1HPGDMAPTSMN1; SMN2LMNA
SCHEMBL5727371 0.79 PDE3B (0.53) ALDH1A1KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL30402755 0.79 HCRTR1 (1.00) HCRTR1ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL2161594 0.79 HCRTR1 (1.00) HCRTR1ALDH1A1KDM4EHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1072655-C New heterocyclic aminomethyl compounds, process for preparing them and pharmaceutical compositions containing them ADIR (FR) 2001-10-10 CN disclosed
EP-0841330-B1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-27 EP disclosed
US-5919784-A ANXIETY, DEPRESSION ADIR ET COMPAGNIE (FR) 1999-07-06 US disclosed
CN-1182083-A New heterocyclic aminomethyl compounds, process for preparing them and pharmaceutical compositions containing them ADIR (FR) 1998-05-20 CN disclosed
EP-0841330-A1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-05-13 EP disclosed