SCHEMBL7768189

SCHEMBL7768189

O=C(c1ccc(OCCN2CCCC2)cc1)c1c(-c2ccc(OCCN3CCCC3)cc2)sc2c(F)c(O)ccc12

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR5A2 O00482 1/20 0.78
ESR1 P03372 19/20 0.71
ESR2 Q92731 18/20 0.71
MEN1 O00255 2/20 0.66
ALDH1A1 P00352 2/20 0.66
LMNA P02545 2/20 0.66
TP53 P04637 2/20 0.66
CYP3A4 P08684 2/20 0.66
MAPT P10636 2/20 0.66
ALOX15 P16050 2/20 0.66
KMT2A Q03164 2/20 0.66
HSD17B10 Q99714 2/20 0.66
TDP1 Q9NUW8 2/20 0.66
PLD2 O14939 1/20 0.66
KDM1A O60341 1/20 0.66
NR1I2 O75469 1/20 0.66
USP2 O75604 1/20 0.66
C5 P01031 1/20 0.66
FYN P06241 1/20 0.66
PGR P06401 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6836618 0.96 NR5A2 (0.85) NR5A2ESR1ESR2MEN1ALDH1A1
SCHEMBL7772161 0.88 ESR1 (0.70) NR5A2ESR1ESR2MEN1ALDH1A1
SCHEMBL7622271 0.88 NR5A2 (1.00) NR5A2ESR1ESR2MEN1ALDH1A1
SCHEMBL7442098 0.86 ESR1 (0.85) NR5A2ESR1ESR2MEN1ALDH1A1
SCHEMBL7768195 0.86 ESR1 (0.67) NR5A2ESR1ESR2MEN1ALDH1A1
SCHEMBL18326547 0.85 NR5A2 (0.79) NR5A2ESR1ESR2MEN1ALDH1A1
SCHEMBL18326522 0.85 NR5A2 (0.85) NR5A2ESR1ESR2MEN1ALDH1A1
SCHEMBL6596230 0.83 ESR1 (0.93) ESR1ESR2MEN1ALDH1A1LMNA
SCHEMBL7452137 0.82 F2 (0.62) NR5A2ESR1ESR2
SCHEMBL6595498 0.81 ESR1 (0.98) ESR1ESR2MEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
US-6025382-A Antithrombotic diamines ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed