SCHEMBL7768296

SCHEMBL7768296

COc1cc(C(=O)c2c(-c3ccc(OCCN4CCCC4)cc3)sc3ccccc23)ccc1CN1CCOCC1

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 18/20 0.71
ESR2 Q92731 18/20 0.71
F2 P00734 1/20 0.62
UBE2N P61088 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6597094 0.91 ESR1 (0.72) ESR1ESR2F2UBE2N
SCHEMBL6596715 0.90 ESR1 (0.60) ESR1ESR2F2
SCHEMBL7775991 0.89 ESR1 (0.55) ESR1ESR2F2
SCHEMBL6592800 0.89 ESR1 (0.82) ESR1ESR2F2UBE2N
SCHEMBL7774305 0.87 ESR1 (0.79) ESR1ESR2UBE2N
SCHEMBL6593201 0.87 ESR1 (0.68) ESR1ESR2F2
SCHEMBL11547737 0.87 ESR1 (0.83) ESR1ESR2F2UBE2N
SCHEMBL6596227 0.87 ESR1 (0.83) ESR1ESR2F2UBE2N
SCHEMBL7414713 0.86 ESR1 (0.73) ESR1ESR2F2
SCHEMBL6596053 0.86 ESR1 (0.79) ESR1ESR2F2UBE2N

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
US-6025382-A Antithrombotic diamines ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed