SCHEMBL7773802

SCHEMBL7773802

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCNC(=O)CN)ccc1NC(=O)c1ccccc1OCCCN

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 2/20 0.40
HTT P42858 2/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HDAC3 O15379 3/20 0.40
HDAC1 Q13547 3/20 0.40
HSP90AA1 P07900 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KCNMA1 Q12791 2/20 0.39
BRD4 O60885 4/20 0.39
BRPF1 P55201 1/20 0.38
PYGL P06737 1/20 0.37
F10 P00742 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7344052 0.99 TP53 (0.40) TP53GAAMAPTHTTLMNA
SCHEMBL7338389 0.96 HDAC3 (0.41) TP53GAAMAPTHTTLMNA
Hydrochloric Acid SCHEMBL7773823 0.95 HDAC3 (0.41) TP53GAAMAPTHTTLMNA
SCHEMBL7339638 0.93 BRD4 (0.43) TP53GAAMAPTHTTLMNA
SCHEMBL7335007 0.93 TP53 (0.41) TP53GAAMAPTHTTLMNA
Hydrochloric Acid SCHEMBL7335902 0.93 TP53 (0.41) TP53GAAMAPTHTTLMNA
Hydrochloric Acid SCHEMBL7346913 0.93 BRD4 (0.42) TP53GAAMAPTHTTLMNA
SCHEMBL7337957 0.92 TP53 (0.46) TP53GAAMAPTHTTLMNA
SCHEMBL7337781 0.92 TP53 (0.47) TP53GAAMAPTHTTLMNA
SCHEMBL7336690 0.92 TP53 (0.40) TP53GAAMAPTHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-B1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2001-09-05 EP disclosed
US-6054457-A Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-25 US disclosed