SCHEMBL7774131

SCHEMBL7774131

CN(C)c1cc(C(=O)c2c(N(C)C)sc3cc(OCc4ccccc4)ccc23)ccc1CN1CCCC1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.43
ESR1 P03372 9/20 0.42
ESR2 Q92731 9/20 0.42
EGFR P00533 2/20 0.41
S1PR1 P21453 1/20 0.41
S1PR5 Q9H228 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6176533 0.92 S1PR1 (0.49) HRH3ESR1ESR2S1PR1S1PR5
SCHEMBL7772387 0.91 ESR1 (0.42) HRH3ESR1ESR2EGFRS1PR1
SCHEMBL6598084 0.91 S1PR1 (0.48) HRH3ESR1ESR2S1PR1S1PR5
SCHEMBL6171046 0.90 CD274 (0.44) ESR1ESR2
SCHEMBL7772159 0.88 CA12 (0.42) HRH3ESR1ESR2EGFR
SCHEMBL7768108 0.86 ESR1 (0.61) ESR1ESR2
SCHEMBL6171041 0.84 ESR1 (0.61) ESR1ESR2
SCHEMBL7447753 0.84 MEN1 (0.44) HRH3ESR1ESR2
SCHEMBL6171651 0.83 EGFR (0.42) HRH3ESR1ESR2EGFR
SCHEMBL6595249 0.79 EGFR (0.43) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed