SCHEMBL7780144

SCHEMBL7780144

CCOC(=O)C=Cc1[nH]c(C(c2ccccc2)(c2ccccc2)c2ccccc2)nc1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
PTGS2 P35354 1/20 0.39
MAPT P10636 8/20 0.39
KDM4E B2RXH2 2/20 0.39
P2RY12 Q9H244 1/20 0.38
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
TTR P02766 1/20 0.38
DPP4 P27487 1/20 0.38
ALOX5 P09917 1/20 0.38
LMNA P02545 3/20 0.37
MDM2 Q00987 2/20 0.37
MDM4 O15151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7412279 0.88 PDE4B (0.41) NPC1RAB9ACA12CA1CA2
SCHEMBL7782729 0.85 HDAC3 (0.38) NPC1RAB9ACA1CA2KDM4E
SCHEMBL7537360 0.75 ERN1 (0.33) NPC1RAB9AKDM4ELMNAALDH1A1
SCHEMBL9267225 0.72 KDM4E (0.46) NPC1RAB9ACA12CA1CA2
SCHEMBL15758898 0.72 KDM4E (0.46) NPC1RAB9ACA12CA1CA2
Ethyl Cinnamate SCHEMBL112446 0.68 CA12 (0.72) NPC1RAB9ACA12CA1CA2
Ethyl Cinnamate SCHEMBL112445 0.68 CA12 (0.72) NPC1RAB9ACA12CA1CA2
Ethyl Cinnamate SCHEMBL12001792 0.68 CA12 (0.72) NPC1RAB9ACA12CA1CA2
Ethyl Cinnamate SCHEMBL1866942 0.68 CA12 (0.72) NPC1RAB9ACA12CA1CA2
SCHEMBL8481698 0.68 MAPT (0.47) NPC1RAB9ACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1135377-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2001-09-26 EP disclosed
WO-2000034254-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2000-06-15 WO disclosed