SCHEMBL7782228

SCHEMBL7782228

CCC[C@@H](C=O)NC(=O)c1cccc(NS(=O)(=O)c2ccc3ccccc3c2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.50
ALDH1A1 P00352 2/20 0.48
LMNA P02545 1/20 0.48
GAA P10253 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
KAT6A Q92794 6/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
AR P10275 1/20 0.47
GGPS1 O95749 1/20 0.46
PLAU P00749 2/20 0.46
GPR27 Q9NS67 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7782230 1.00 AKR1C3 (0.50) AKR1C3ALDH1A1LMNAGAASMN1; SMN2
SCHEMBL7787806 0.92 AKR1C3 (0.52) AKR1C3ALDH1A1LMNAGAASMN1; SMN2
SCHEMBL7787778 0.90 AKR1C3 (0.47) AKR1C3ALDH1A1LMNAGAASMN1; SMN2
SCHEMBL7782218 0.86 AKR1C3 (0.53) AKR1C3ALDH1A1LMNAGAASMN1; SMN2
SCHEMBL7782219 0.86 AKR1C3 (0.53) AKR1C3ALDH1A1LMNAGAASMN1; SMN2
SCHEMBL7790030 0.85 AKR1C3 (0.51) AKR1C3ALDH1A1LMNAGAASMN1; SMN2
SCHEMBL7790027 0.85 AKR1C3 (0.51) AKR1C3ALDH1A1LMNAGAASMN1; SMN2
SCHEMBL7791348 0.82 AKR1C3 (0.46) AKR1C3ALDH1A1LMNAGAASMN1; SMN2
SCHEMBL7791346 0.82 AKR1C3 (0.46) AKR1C3ALDH1A1LMNAGAASMN1; SMN2
SCHEMBL7787817 0.81 AKR1C3 (0.53) AKR1C3ALDH1A1LMNAGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed
CN-1238761-A benzamide aldehydes and their use as cysteine protease inhibitors BASF AG (DE) 1999-12-15 CN disclosed