SCHEMBL7784843

SCHEMBL7784843

COC(=O)CC(S)CC(=O)OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.50
HSD17B10 Q99714 2/20 0.50
MGAM O43451 2/20 0.43
GAA P10253 2/20 0.43
SI P14410 2/20 0.43
MGAM2 Q2M2H8 2/20 0.43
HSP90AB1 P08238 1/20 0.37
KMT2A Q03164 2/20 0.36
TET2 Q6N021 1/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 2/20 0.34
CA12 O43570 1/20 0.34
CA14 Q9ULX7 1/20 0.34
KDM4E B2RXH2 1/20 0.34
RECQL P46063 1/20 0.34
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34
MAPT P10636 3/20 0.34
RAB9A P51151 1/20 0.34
MMP1 P03956 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5898819 0.87
SCHEMBL8399384 0.84 TSHR (0.50) TSHRHSD17B10MGAMGAASI
SCHEMBL5898807 0.84 TSHR (0.41) TSHRHSD17B10MGAMGAASI
SCHEMBL14239656 0.83 TSHR (0.50) TSHRHSD17B10MGAMGAASI
SCHEMBL690378 0.81
SCHEMBL5898830 0.81
SCHEMBL8499849 0.81
SCHEMBL9876817 0.79 TSHR (0.46) TSHRHSD17B10MGAMGAASI
SCHEMBL11804805 0.79 ZDHHC7 (0.46) HSD17B10KMT2AMEN1LMNARECQL
SCHEMBL7631058 0.77 TSHR (0.44) TSHRHSD17B10MGAMGAASI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070087-B1 INTERMEDIATES FOR THE SYNTHESIS OF CYCLIC P1 LINKERS AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2019-04-10 EP disclosed
EP-1142881-A1 POLY(ADP-RIBOSE) POLYMERASE INHIBITORS CONSISTING OF PYRIMIDINE DERIVATIVES MEIJI SEIKA KAISHA LTD. (JP) 2001-10-10 EP disclosed
US-4242518-A Thiophene compounds and their manufacture BASF AKTIENGESELLSCHAFT (DE) 1980-12-30 US disclosed
US-4239897-A Thiophene compounds and their manufacture BASF AKTIENGESELLSCHAFT (DE) 1980-12-16 US disclosed