SCHEMBL7790862

SCHEMBL7790862

O=C(NC(CO)Cc1c[nH]c2ccccc12)c1cccc(NS(=O)(=O)c2ccc3ccccc3c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
HTT P42858 3/20 0.52
MAPT P10636 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
LMNA P02545 1/20 0.52
HDAC8 Q9BY41 4/20 0.50
HDAC6 Q9UBN7 4/20 0.50
HDAC2 Q92769 3/20 0.50
MMP9 P14780 2/20 0.47
MMP1 P03956 1/20 0.47
MMP2 P08253 1/20 0.47
MMP3 P08254 1/20 0.47
MMP7 P09237 1/20 0.47
MMP14 P50281 1/20 0.47
ALDH1A1 P00352 2/20 0.47
HTR6 P50406 7/20 0.47
CCKBR P32239 1/20 0.46
HDAC3 O15379 2/20 0.45
HDAC4 P56524 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7782244 0.87 HDAC8 (0.49) MEN1KMT2AHTTMAPTSMN1; SMN2
SCHEMBL7791333 0.83 AKR1C3 (0.54) MEN1KMT2AHTTMAPTSMN1; SMN2
SCHEMBL7791335 0.83 AKR1C3 (0.54) MEN1KMT2AHTTMAPTSMN1; SMN2
SCHEMBL7787817 0.81 AKR1C3 (0.53) MEN1KMT2ASMN1; SMN2LMNAHDAC8
SCHEMBL7790027 0.79 AKR1C3 (0.51) MEN1KMT2ASMN1; SMN2LMNAHDAC8
SCHEMBL7790030 0.79 AKR1C3 (0.51) MEN1KMT2ASMN1; SMN2LMNAHDAC8
SCHEMBL13902824 0.77 MEN1 (0.61) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL7786978 0.77 AKR1C3 (0.48) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL7786983 0.77 AKR1C3 (0.48) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL5149228 0.77 MEN1 (0.66) MEN1KMT2AHDAC8HDAC6HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed