SCHEMBL7791357

SCHEMBL7791357

COc1ccc(C=Cc2ccccc2C(=O)NC(CO)Cc2ccccc2)cc1OC

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 9/20 0.75
CTSB P07858 5/20 0.52
CTSL P07711 2/20 0.52
ROCK2 O75116 3/20 0.51
ROCK1 Q13464 3/20 0.51
ALDH1A1 P00352 5/20 0.48
TAS1R3 Q7RTX0 1/20 0.48
TAS1R1 Q7RTX1 1/20 0.48
CTSS P25774 2/20 0.48
CTSK P43235 2/20 0.48
CYP1A2 P05177 2/20 0.47
CYP1A1 P04798 1/20 0.47
CYP19A1 P11511 1/20 0.47
CYP1B1 Q16678 1/20 0.47
HPGD P15428 2/20 0.46
HTT P42858 1/20 0.46
KDM4E B2RXH2 3/20 0.46
POLB P06746 1/20 0.46
PKM P14618 1/20 0.46
TTR P02766 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7791353 1.00 CAPN1 (0.75) CAPN1CTSBCTSLROCK2ROCK1
SCHEMBL7787053 0.86 CAPN1 (1.00) CAPN1CTSBCTSLALDH1A1TAS1R3
SCHEMBL7787056 0.86 CAPN1 (1.00) CAPN1CTSBCTSLALDH1A1TAS1R3
SCHEMBL7791345 0.84 CAPN1 (0.70) CAPN1CTSBCTSLROCK2ROCK1
SCHEMBL7789913 0.83 CAPN1 (0.74) CAPN1CTSBCTSLROCK2ROCK1
SCHEMBL7789911 0.83 CAPN1 (0.74) CAPN1CTSBCTSLROCK2ROCK1
SCHEMBL7694680 0.80 CAPN1 (0.72) CAPN1CTSBCTSLALDH1A1TAS1R3
SCHEMBL1930485 0.80 CAPN1 (0.60) CAPN1CTSBCTSLROCK2ROCK1
SCHEMBL1930486 0.80 CAPN1 (0.60) CAPN1CTSBCTSLROCK2ROCK1
SCHEMBL7695839 0.79 CAPN1 (0.70) CAPN1CTSBCTSLALDH1A1TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed