SCHEMBL7795324

SCHEMBL7795324

CN1c2ccccc2C(C(=O)Oc2cc(Cl)c(Cl)cc2Cl)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
FABP7 O15540 1/20 0.47
FABP3 P05413 1/20 0.47
FABP5 Q01469 1/20 0.47
EGFR P00533 2/20 0.39
SRC P12931 1/20 0.39
KMT2A Q03164 4/20 0.37
L3MBTL1 Q9Y468 4/20 0.37
MEN1 O00255 3/20 0.37
GAA P10253 3/20 0.37
LMNA P02545 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAPT P10636 2/20 0.36
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 3/20 0.34
TSHR P16473 2/20 0.34
GLA P06280 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8741648 0.83 FABP3 (0.48) HDAC4HDAC7HDAC5FABP3EGFR
SCHEMBL7796561 0.81 FABP7 (0.38) HDAC4HDAC7HDAC5FABP7FABP3
SCHEMBL31613805 0.81 HDAC4 (0.48) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL5665136 0.81 HDAC4 (0.48) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL7795339 0.79 HDAC4 (0.51) HDAC4HDAC7HDAC5FABP7FABP3
SCHEMBL13005786 0.79 HDAC4 (0.51) HDAC4HDAC7HDAC5FABP7FABP3
SCHEMBL8741687 0.79 HDAC4 (0.51) HDAC4HDAC7HDAC5FABP7FABP3
SCHEMBL13005780 0.78 HDAC4 (0.57) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL8741803 0.78 HDAC4 (0.50) HDAC4HDAC7HDAC5FABP7FABP3
SCHEMBL8741624 0.78 HDAC4 (0.50) HDAC4HDAC7HDAC5EGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750748-B1 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN INC (US) 2001-12-05 EP claimed
US-5750698-A USEFUL IN DETECTING BOTH PEROXIDASE AND PEROXIDE LUMIGEN, INC. (US) 1998-05-12 US claimed
WO-1995023971-A1 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1995-09-08 WO claimed
EP-0750748-B1 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN INC (US) 2001-12-05 EP disclosed
US-5750698-A USEFUL IN DETECTING BOTH PEROXIDASE AND PEROXIDE LUMIGEN, INC. (US) 1998-05-12 US disclosed
US-5593845-A BY REACTION WITH PEROXIDES AND PEROXIDASE; DETECTION OF HAPTENS, PROTEINS, ANTIBODIES IN ENZYME IMMUNOASSAY LUMIGEN, INC. (US) 1997-01-14 US disclosed
WO-1995023971-A1 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1995-09-08 WO disclosed