SCHEMBL7806754

SCHEMBL7806754

COC(=O)N[C@H](C(=O)N1Cc2ccccc2CC1C(=O)O)C(C)C

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACE P12821 8/20 0.59
ABCB11 O95342 1/20 0.51
FNTA P49354 1/20 0.47
FNTB P49356 1/20 0.47
PGGT1B P53609 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9545015 0.90 ACE (0.56) ACEABCB11FNTAFNTBPGGT1B
SCHEMBL27726228 0.90 ACE (0.56) ACEABCB11FNTAFNTBPGGT1B
SCHEMBL27726229 0.90 ACE (0.56) ACEABCB11FNTAFNTBPGGT1B
SCHEMBL9545013 0.90 ACE (0.56) ACEABCB11FNTAFNTBPGGT1B
SCHEMBL3728963 0.84 XIAP (0.61) ACE
SCHEMBL15569217 0.84 XIAP (0.61) ACE
SCHEMBL29670215 0.83 ACE (0.51) ACEABCB11
SCHEMBL27726218 0.82 ACE (0.55) ACEABCB11POLB
SCHEMBL27726298 0.82 HDAC8 (0.52) ACEFNTAFNTBPGGT1B
SCHEMBL27726215 0.82 ACE (0.55) ACEABCB11POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1114822-A2 Indoles and tetrahydroisoquinolines containing alpha-keto oxadiazoles as serine protease inhibitors Cortech Inc. (US) 2001-07-11 EP disclosed
US-6100238-A USEFUL AS INHIBITORS OF HUMAN NEUTROPHIL ELASTASE (HNE) FOR THE TREATMENT OF HNE-MEDIATED PROCESSES IMPLICATED IN CONDITIONS SUCH AS ADULT RESPIRATORY DISTRESS SYNDROME, SEPTIC SHOCK AND MULTIPLE ORGAN FAILURE CORTECH INC. (US) 2000-08-08 US disclosed