SCHEMBL7808149

SCHEMBL7808149

OCc1ccc2cc(Cl)ccc2n1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.49
HDAC2 Q92769 2/20 0.49
S1PR4 O95977 2/20 0.47
CCR1 P32246 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
MCHR1 Q99705 1/20 0.45
FAAH O00519 1/20 0.44
PDE10A Q9Y233 1/20 0.43
HTR3A P46098 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
ALDH1A1 P00352 1/20 0.40
BACE1 P56817 1/20 0.40
CYP2A6 P11509 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
NOTUM Q6P988 3/20 0.39
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7809623 0.86 S1PR4 (0.49) HDAC1HDAC2S1PR4CCR1TDP1
SCHEMBL2412433 0.82 HDAC1 (0.47) HDAC1HDAC2FAAHPDE10AHTR3A
SCHEMBL9022559 0.81 PDE10A (0.46) HDAC1HDAC2FAAHPDE10AHTR3A
SCHEMBL201434 0.81 CCR1 (0.47) HDAC1HDAC2CCR1TDP1FAAH
SCHEMBL5103462 0.81 HDAC1 (0.46) HDAC1HDAC2FAAHPDE10AHTR3A
SCHEMBL4720632 0.79 HDAC1 (0.51) HDAC1HDAC2FAAHPDE10AALDH1A1
SCHEMBL27529644 0.78 PDE10A (0.47) HDAC1HDAC2FAAHPDE10AHTR3A
SCHEMBL14127821 0.78 PDE10A (0.50) HDAC1HDAC2MCHR1FAAHPDE10A
SCHEMBL31434472 0.78 HDAC1 (0.50) HDAC1HDAC2FAAHPDE10AHTR3A
SCHEMBL12516193 0.77 CCR1 (0.47) HDAC1HDAC2CCR1MCHR1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0685478-B1 QUINOLINE DERIVATIVES UBE INDUSTRIES (JP) 2001-10-24 EP disclosed
CN-1046279-C Quinoline derivative UBE INDUSTRIES (JP) 1999-11-10 CN disclosed
US-5591752-A LEUKOTRIENE ANTAGONIST, ANTIALLERGEN, ANTIINFLAMMATORY AGENT, DIBENZ(B,E)OXEPINE UBE INDUSTRIES, LTD. (JP) 1997-01-07 US disclosed
EP-0685478-A1 QUINOLINE DERIVATIVE UBE INDUSTRIES, LTD. (JP) 1995-12-06 EP disclosed