SCHEMBL7808663

SCHEMBL7808663

OCc1nc2ccc(Sc3ncc[nH]3)cc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.50
NPSR1 Q6W5P4 1/20 0.46
GCK P35557 1/20 0.38
CBFB Q13951 1/20 0.37
RAD52 P43351 1/20 0.36
RHEB Q15382 1/20 0.36
KMT2A Q03164 3/20 0.35
POLB P06746 1/20 0.35
TPSAB1 Q15661 3/20 0.35
PRSS1 P07477 2/20 0.35
F2 P00734 1/20 0.35
F10 P00742 1/20 0.35
PLG P00747 1/20 0.35
PLAU P00749 1/20 0.35
PRSS2 P07478 1/20 0.35
PRSS3 P35030 1/20 0.35
RAB9A P51151 1/20 0.35
PKM P14618 3/20 0.35
CHEK1 O14757 1/20 0.35
PRKD3 O94806 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8479187 0.99 TDP1 (0.49) TDP1NPSR1GCKCBFBRAD52
SCHEMBL7808661 0.91 TDP1 (0.43) TDP1NPSR1GCKRHEBKMT2A
Hydrochloric Acid SCHEMBL8479183 0.90 TDP1 (0.42) TDP1NPSR1GCKRAD52RHEB
SCHEMBL7808593 0.80 TDP1 (0.54) TDP1NPSR1RAD52KMT2APOLB
Hydrochloric Acid SCHEMBL8480485 0.78 TDP1 (0.52) TDP1NPSR1RAD52KMT2APOLB
SCHEMBL7808619 0.78 TDP1 (0.52) TDP1NPSR1CBFBRHEBKMT2A
Hydrochloric Acid SCHEMBL8479272 0.77 TDP1 (0.51) TDP1NPSR1CBFBRAD52KMT2A
Hydrochloric Acid SCHEMBL8477383 0.74 TDP1 (0.48) TDP1NPSR1RAD52KMT2APOLB
SCHEMBL12635706 0.72 TDP1 (0.55) TDP1NPSR1RAD52KMT2APOLB
SCHEMBL7809674 0.69 TDP1 (0.40) TDP1NPSR1CBFBDYRK1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820990-B1 Benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR (FR) 2001-01-17 EP disclosed
EP-0820990-A2 Novel benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR ET COMPAGNIE (FR) 1998-01-28 EP disclosed