SCHEMBL7810280

SCHEMBL7810280

O=CCC1(c2ccc(Cl)c(Cl)c2)CCC(=O)NC1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 20/20 0.47
SLC6A3 Q01959 19/20 0.47
SLC6A2 P23975 12/20 0.40
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7811639 0.82 SLC6A4 (0.61) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL6543319 0.79 SLC6A4 (0.45) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL5901153 0.78 SLC6A4 (0.43) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL27528569 0.78 SLC6A4 (0.43) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL7371366 0.77 SLC6A4 (0.63) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL5086634 0.76 SLC6A4 (0.64) SLC6A4SLC6A3SLC6A2
SCHEMBL6543222 0.75 SLC6A4 (0.46) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL7811794 0.75 SLC6A4 (0.44) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL6999461 0.73 SLC6A4 (0.41) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL6956287 0.72 TACR1 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775132-B1 (AZETIDIN-1-YLALKYL)LACTAMS AS TACHYKININ ANTAGONISTS PFIZER LTD (GB) 2001-03-28 EP disclosed
US-5968923-A ANTIINFLAMMATORY AGENTS, TREATMENT OF NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS PFIZER INC. (US) 1999-10-19 US disclosed
WO-1996005193-A1 (AZETIDIN-1-YLALKYL)LACTAMS AS TACHYKININ ANTAGONISTS PFIZER LIMITED (GB) 1996-02-22 WO disclosed