SCHEMBL7811237

SCHEMBL7811237

COc1ccc(COc2ccc3[nH]c(CO)nc3c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.54
RAB9A P51151 4/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
TP53 P04637 2/20 0.51
ALDH1A1 P00352 1/20 0.51
MAOB P27338 4/20 0.46
MAOA P21397 2/20 0.46
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
GAA P10253 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.45
RHEB Q15382 3/20 0.45
CBFB Q13951 1/20 0.44
APP P05067 3/20 0.43
FLT3 P36888 1/20 0.43
CYP2E1 P05181 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C8 P10632 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7811241 0.90 MAOB (0.58) NPC1RAB9ASMN1; SMN2TP53ALDH1A1
SCHEMBL4470392 0.88 NPC1 (0.52) NPC1RAB9ASMN1; SMN2TP53ALDH1A1
SCHEMBL1050471 0.87 NPC1 (0.52) NPC1RAB9ASMN1; SMN2TP53ALDH1A1
SCHEMBL7806914 0.87 NPC1 (0.45) NPC1RAB9ASMN1; SMN2TP53ALDH1A1
Hydrochloric Acid SCHEMBL8474019 0.86 NPC1 (0.44) NPC1RAB9ASMN1; SMN2TP53ALDH1A1
SCHEMBL7811234 0.83 GRIN1 (0.49) NPC1RAB9ASMN1; SMN2TP53ALDH1A1
SCHEMBL2019822 0.81 NPC1 (0.49) NPC1RAB9ASMN1; SMN2TP53ALDH1A1
SCHEMBL7806919 0.76 MAOB (0.55) NPC1RAB9ASMN1; SMN2TP53MAOB
SCHEMBL9598328 0.76 CYP2D6 (0.48) NPC1RAB9ASMN1; SMN2TP53ALDH1A1
SCHEMBL31284816 0.76 F10 (0.61) NPC1RAB9ASMN1; SMN2TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820990-B1 Benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR (FR) 2001-01-17 EP disclosed
EP-0820990-A2 Novel benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR ET COMPAGNIE (FR) 1998-01-28 EP disclosed