SCHEMBL7811779

SCHEMBL7811779

c1ccc2sc(C3CC[N]3)cc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.47
DRD2 P14416 1/20 0.47
SLC6A3 Q01959 4/20 0.41
SLC6A2 P23975 2/20 0.41
ALOX5 P09917 1/20 0.41
CHRM2 P08172 2/20 0.39
CHRM4 P08173 2/20 0.39
CHRM5 P08912 2/20 0.39
CHRM1 P11229 2/20 0.39
CHRM3 P20309 2/20 0.39
CYP2A6 P11509 3/20 0.38
ASIC3 Q9UHC3 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38
MGLL Q99685 1/20 0.38
KDM1A O60341 1/20 0.38
BCL2L1 Q07817 1/20 0.37
SIGMAR1 Q99720 3/20 0.37
CA2 P00918 1/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7716348 0.87 SLC6A4 (0.43) SLC6A4DRD2SLC6A3SLC6A2ALOX5
SCHEMBL28359596 0.79 SLC6A4 (0.61) SLC6A4DRD2SLC6A3SLC6A2ALOX5
SCHEMBL31172103 0.79 SLC6A4 (0.61) SLC6A4DRD2SLC6A3SLC6A2ALOX5
SCHEMBL4670974 0.79 SLC6A4 (0.54) SLC6A4DRD2SLC6A3SLC6A2ALOX5
SCHEMBL6752313 0.78 SLC6A4 (0.38) SLC6A4DRD2SLC6A3SLC6A2ALOX5
SCHEMBL5744613 0.78 SLC6A4 (0.38) SLC6A4DRD2SLC6A3SLC6A2ALOX5
SCHEMBL20172556 0.72 SLC6A4 (0.39) SLC6A4DRD2SLC6A3SLC6A2ALOX5
SCHEMBL29261831 0.72 SLC6A4 (0.46) SLC6A4DRD2SLC6A3SLC6A2ALOX5
SCHEMBL2708963 0.71 SLC6A4 (0.54) SLC6A4DRD2SLC6A3SLC6A2ALOX5
SCHEMBL14559225 0.70 SLC6A4 (0.38) SLC6A4DRD2SLC6A3SLC6A2ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0873340-B1 HETEROCYCLIC SUBSTITUTED CYCLOPENTANE COMPOUNDS ABBOTT LAB (US) 2001-11-21 EP disclosed
US-6143749-A Heterocyclic substituted cyclopentane compounds ABBOTT LABORATORIES (US) 2000-11-07 US disclosed
US-5665721-A ADENOSINE KINASE INHIBITORS ABBOTT LABORATORIES (US) 1997-09-09 US disclosed