SCHEMBL7812899

SCHEMBL7812899

O=C1CC(c2ccc(F)cc2)CCN1Cc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.59
TSHR P16473 1/20 0.59
HTT P42858 1/20 0.51
KCNH2 Q12809 1/20 0.51
GRIN2B Q13224 1/20 0.51
PDE4A P27815 1/20 0.47
PDE4B Q07343 1/20 0.47
PDE4C Q08493 1/20 0.47
PDE4D Q08499 1/20 0.47
CHRM4 P08173 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581697 1.00 HPGD (0.59) HPGDTSHRHTTKCNH2GRIN2B
SCHEMBL28169051 0.84 TP53 (0.50) HTTKCNH2GRIN2B
SCHEMBL28298576 0.83 PDE4A (0.56) HPGDTSHRPDE4APDE4BPDE4C
SCHEMBL3038179 0.77 HPGD (0.56) HPGDTSHRGRIN2BCHRM4
SCHEMBL24791557 0.76 PDE4A (0.48) HPGDTSHRPDE4APDE4BPDE4C
SCHEMBL9563914 0.76 HPGD (0.52) HPGDTSHRPDE4APDE4BPDE4C
SCHEMBL16033027 0.75 HPGD (1.00) HPGDTSHRPDE4APDE4BPDE4C
SCHEMBL12563130 0.75 KCNH2 (0.47) KCNH2GRIN2B
SCHEMBL2794992 0.74 HTT (0.44) HTTKCNH2GRIN2B
SCHEMBL11123316 0.74 HPGD (0.53) HPGDTSHRGRIN2BCHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986389-A4 NOVEL PROCESS SMITHKLINE BEECHAM CORP (US) 2001-09-12 EP disclosed
EP-0986389-A1 NOVEL PROCESS SMITHKLINE BEECHAM CORPORATION (US) 2000-03-22 EP disclosed
WO-1998053824-A1 NOVEL PROCESS SMITHKLINE BEECHAM CORPORATION (US) 1998-12-03 WO disclosed