SCHEMBL7817862

SCHEMBL7817862

CC(C)C(O)(c1ccc2cc(N(C)C(N)=O)ccc2c1)c1c[nH]cn1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 17/20 0.43
CYP3A4 P08684 16/20 0.43
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4025856 0.82 CYP17A1 (0.64) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL5752821 0.80 CYP17A1 (0.62) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL5750907 0.79 CYP3A4 (0.44) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL5753882 0.79 CYP3A4 (0.44) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL4027619 0.79 CYP3A4 (0.51) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL5750604 0.79 CYP17A1 (0.50) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL5752256 0.78 CYP3A4 (0.44) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL5751835 0.78 CYP3A4 (0.44) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL5754667 0.78 CYP17A1 (0.51) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL5753350 0.78 CYP3A4 (0.53) CYP17A1CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073640-A1 NAPHTHALENE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2001-02-07 EP disclosed
WO-1999054309-A1 NAPHTHALENE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-10-28 WO disclosed