SCHEMBL7818751

SCHEMBL7818751

CN(C)C(=O)c1cccc(-c2ccc3c(nnn3CC3CC3)c2Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 9/20 0.47
CECR2 Q9BXF3 2/20 0.47
BRD4 O60885 6/20 0.44
FYN P06241 1/20 0.41
EP300 Q09472 1/20 0.39
CREBBP Q92793 1/20 0.39
TDO2 P48775 1/20 0.39
PTGER4 P35408 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3476569 0.87 GRM2 (0.53) GRM2FYNTDO2
SCHEMBL7808009 0.86 GRM2 (0.47) GRM2BRD4EP300CREBBPTDO2
SCHEMBL7816317 0.81 GRM2 (0.47) GRM2TDO2PTGER4
SCHEMBL3473877 0.80 GRM2 (0.53) GRM2BRD4CREBBPTDO2
SCHEMBL3476934 0.79 GRM2 (0.55) GRM2TDO2
SCHEMBL3475682 0.79 GRM2 (0.50) GRM2CREBBPTDO2
SCHEMBL3476594 0.79 GRM2 (0.52) GRM2TDO2
SCHEMBL7816041 0.79 GRM2 (0.59) GRM2TDO2
SCHEMBL3475606 0.77 GRM2 (0.49) GRM2TDO2PTGER4
SCHEMBL3478502 0.77 GRM2 (0.50) GRM2BRD4TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO disclosed