Teloxantrone

Teloxantrone

SCHEMBL782387

CNCCNc1ccc2c3c(nn2CCNCCO)-c2c(O)ccc(O)c2C(=O)c13

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 2/20 0.70
MEN1 O00255 2/20 0.54
USP2 O75604 2/20 0.54
LMNA P02545 2/20 0.54
TP53 P04637 2/20 0.54
MAPK1 P28482 2/20 0.54
RECQL P46063 2/20 0.54
BLM P54132 2/20 0.54
KMT2A Q03164 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
NSD2 O96028 2/20 0.54
CSNK2A1 P68400 2/20 0.54
NPC1 O15118 1/20 0.54
SLC22A2 O15244 1/20 0.54
SLC22A1 O15245 1/20 0.54
CACNA1F O60840 1/20 0.54
SLC22A3 O75751 1/20 0.54
EGFR P00533 1/20 0.54
ESR1 P03372 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Teloxantrone SCHEMBL9177269 0.99 TOP2A (0.69) TOP2AMEN1USP2LMNATP53
Teloxantrone SCHEMBL3195 0.98 TOP2A (0.68) TOP2AMEN1USP2LMNATP53
Teloxantrone SCHEMBL29397399 0.98 TOP2A (0.68) TOP2AMEN1USP2LMNATP53
SCHEMBL10804721 0.96 TOP2A (0.70) TOP2AMEN1USP2LMNATP53
SCHEMBL10998300 0.94 TOP2A (0.79) TOP2AMEN1USP2LMNATP53
SCHEMBL10802433 0.91 TOP2A (0.64) TOP2AMEN1USP2LMNATP53
SCHEMBL10805640 0.90 TOP2A (0.70) TOP2AMEN1USP2LMNATP53
SCHEMBL10805304 0.90 TOP2A (0.72) TOP2AMEN1USP2LMNATP53
Piroxantrone SCHEMBL93599 0.90 TOP2A (0.69) TOP2AMEN1USP2LMNATP53
SCHEMBL10803111 0.90 TOP2A (0.72) TOP2AMEN1USP2LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1082 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250275946-A1 COMBINATION THERAPY FOR THE TREATMENT OF CANCER UNM RAINFOREST INNOVATIONS (US) 2025-09-04 US claimed
EP-3441089-B1 TREATMENT METHODS USING ADENOVIRUS VASCULAR BIOGENICS LTD (IL) 2022-12-14 EP claimed
US-20220347108-A1 PROCESS FOR PRODUCING A PHARMACEUTICAL FORMULATION COMPRISING CRYSTALLINE AND AMORPHOUS FRACTIONS OF AN ACTIVE SUBSTANCE BAYER AKTIENGESELLSCHAFT (DE) 2022-11-03 US claimed
WO-2022169634-A9 COMBINATION THERAPY FOR THE TREATMENT OF CANCER UNM RAINFOREST INNOVATIONS (US) 2022-09-22 WO claimed
EP-4041201-A1 PROCESS FOR PRODUCING A PHARMACEUTICAL FORMULATION COMPRISING CRYSTALLINE AND AMORPHOUS FRACTIONS OF AN ACTIVE SUBSTANCE Bayer Aktiengesellschaft (DE) 2022-08-17 EP claimed
WO-2022169634-A1 COMBINATION THERAPY FOR THE TREATMENT OF CANCER UNM RAINFOREST INNOVATIONS (US) 2022-08-11 WO claimed
WO-2021069349-A1 PROCESS FOR PRODUCING A PHARMACEUTICAL FORMULATION COMPRISING CRYSTALLINE AND AMORPHOUS FRACTIONS OF AN ACTIVE SUBSTANCE BAYER AKTIENGESELLSCHAFT (DE) 2021-04-15 WO claimed
EP-3804701-A1 METHOD FOR PREPARING A PHARMACEUTICAL FORMULATION COMPRISING CRYSTALLINE AND AMORPHOUS PORTIONS OF AN ACTIVE SUBSTANCE Bayer AG (DE) 2021-04-14 EP claimed
EP-3804702-A1 METHOD FOR PREPARING A PHARMACEUTICAL FORMULATION COMPRISING ACTIVE AGENT, POLYMER AND SURFACTANT Bayer AG (DE) 2021-04-14 EP claimed
EP-3191114-B1 OCCIDIOFUNGIN FORMULATIONS AND USES THEREOF UNIV MISSISSIPPI STATE (US) 2021-03-03 EP claimed
CN-1634585-A Anti-cancer medicine composition SHANDONG LANJIN BIOENGINEERING (CN) 2005-07-06 CN claimed
CN-1634583-A Anti-cancer medicine composition containing antineoplastic antibiotics SHANDONG LANJIN BIOENGINEERING (CN) 2005-07-06 CN claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
US-20030036794-A1 Coated implantable medical device COOK INCORPORATED 2003-02-20 US claimed
EP-1085891-A1 MULTIBINDING INHIBITORS OF TOPOISOMERASE Advanced Medicine, Inc. (US) 2001-03-28 EP claimed
CN-1261803-A Antioxidant enhancement of therapy for hyperproliferative conditions ATHEROGENICS INC (US) 2000-08-02 CN claimed
WO-1999064054-A9 MULTIBINDING INHIBITORS OF TOPOISOMERASE ADVANCED MEDICINE INC (US) 2000-03-02 WO claimed
WO-1999064054-A1 MULTIBINDING INHIBITORS OF TOPOISOMERASE ADVANCED MEDICINE, INC. (US) 1999-12-16 WO claimed
EP-0103381-B1 SUBSTITUTED ANTHRA(1,9-CD)PYRAZOL-6(2H)-ONES WARNER-LAMBERT COMPANY (US) 1987-09-23 EP claimed
EP-0103381-A1 Substituted anthra(1,9-cd)pyrazol-6(2H)-ones WARNER-LAMBERT COMPANY (US) 1984-03-21 EP claimed