Pixantrone

Pixantrone

SCHEMBL7825

NCCNc1ccc(NCCN)c2c1C(=O)c1ccncc1C2=O

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 1/20 0.72
MUS81 Q96NY9 1/20 0.72
KDM4C Q9H3R0 2/20 0.49
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
CDC25B P30305 1/20 0.45
BLM P54132 5/20 0.43
MAPT P10636 5/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
TP53 P04637 3/20 0.43
CYP3A4 P08684 3/20 0.43
CASP1 P29466 3/20 0.43
CASP7 P55210 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
NSD2 O96028 1/20 0.43
POLB P06746 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
TOP2B Q02880 1/20 0.42
PRKCH P24723 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pixantrone SCHEMBL29372192 1.00 ECE1 (0.72) ECE1MUS81KDM4CMAOAMAOB
Pixantrone SCHEMBL17673194 0.98 ECE1 (0.70) ECE1MUS81KDM4CMAOAMAOB
Pixantrone SCHEMBL7771183 0.98 ECE1 (0.70) ECE1MUS81KDM4CMAOAMAOB
SCHEMBL28381205 0.93 ECE1 (0.65) ECE1MUS81KDM4CMAOAMAOB
SCHEMBL29642348 0.93 ECE1 (0.65) ECE1MUS81KDM4CMAOAMAOB
SCHEMBL28381199 0.93 ECE1 (0.65) ECE1MUS81KDM4CMAOAMAOB
SCHEMBL28378350 0.93 ECE1 (0.65) ECE1MUS81KDM4CMAOAMAOB
SCHEMBL13524774 0.93 ECE1 (0.68) ECE1MUS81KDM4CMAOAMAOB
SCHEMBL29642192 0.93 ECE1 (0.65) ECE1MUS81KDM4CMAOAMAOB
SCHEMBL29642322 0.93 ECE1 (0.65) ECE1MUS81KDM4CMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 14938 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026101236-A1 PEPTIDES SPECIFICALLY BINDING TO CCR8, AND USE THEREOF 경희대학교 산학협력단 2026-05-15 WO claimed
EP-4737898-A2 SEPARATION AND ISOLATION OF NUCLEIC ACIDS USING AFFINITY LIGANDS BOUND TO A SOLID SURFACE EMP Biotech GmbH (DE) 2026-05-06 EP claimed
US-12600696-B2 Aromatic compounds Xeniopro GmbH (DE) 2026-04-14 US claimed
US-20260085061-A1 PHTHALAZINE DERIVATIVES AS PYRUVATE KINASE MODULATORS SITRYX THERAPEUTICS LIMITED (GB) 2026-03-26 US claimed
EP-4692122-A1 HUMANIZED ANTIBODIES TARGETING EPHA10 Korea University Research and Business Foundation (KR) 2026-02-11 EP claimed
US-20260000782-A1 ITGB2-MEDIATED DRUG DELIVERY SYSTEM TWINPIG BIOLAB INC. (KR) 2026-01-01 US claimed
US-20250381202-A1 PRODRUG KIT FOR MULTI-PRONGED CHEMOTHERAPY ZOUNEK ALEX (DE) 2025-12-18 US claimed
US-20250376507-A1 NOVEL TUMOR ANTIGEN-TARGETING ANTICANCER AGENT UNIV NAT CHONNAM IND FOUND (KR) 2025-12-11 US claimed
EP-4640714-A2 METHODS FOR ASSESSING RISK OF DEVELOPING A VIRAL DISEASE USING A GENETIC TEST PML Screening, LLC (US) 2025-10-29 EP claimed
EP-4638443-A1 TRANSIENT RECEPTOR POTENTIAL VANILLOID 6 INHIBITORS Uniquest Pty Limited (AU) 2025-10-29 EP claimed
WO-2001028521-A2 LIPOSOME FORMULATION OF 6,9-BIS-[(2-AMINOETHYL)-AMINO]BENZO[G]ISOQUINOLINE-5,10-DIONE DIMALEATE NOVUSPHARMA S.P.A. (IT) 2001-04-26 WO claimed
EP-0503537-B1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones UNIV VERMONT (US) 1997-05-14 EP claimed
US-5616709-A Method of synthesis for 6,9-bis[(2-aminoethyl)amino]benzo[g]isoquinoline-5,10-dione and its dimaleate salt BOEHRINGER MANNHEIM GMBH (IT) 1997-04-01 US claimed
EP-0752857-A1 AN IMPROVED METHOD OF SYNTHESIS FOR 6,9-BIS (2-AMINOETHYL)AMINO]BENZO g]ISOQUINOLINE-5,10-DIONE AND ITS DIMALEATE SALT BOEHRINGER MANNHEIM ITALIA S.p.A. (IT) 1997-01-15 EP claimed
US-5587382-A ANTITUMOR AGENTS BOEHRINGER MANNHEIM ITALIA, SPA (IT) 1996-12-24 US claimed
US-5506232-A 6,9-bis[(2-aminoethyl)amino]benzo[g]isoquinoline-5,10-dione and its dimaleate salt BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1996-04-09 US claimed
WO-1995026189-A1 AN IMPROVED METHOD OF SYNTHESIS FOR 6,9-BIS[(2-AMINOETHYL)AMINO]BENZO[g]ISOQUINOLINE-5,10-DIONE AND ITS DIMALEATE SALT BOEHRINGER MANNHEIM ITALIA, S.P.A. (US) 1995-10-05 WO claimed
EP-0575526-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1993-12-29 EP claimed
WO-1992015300-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO[g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1992-09-17 WO claimed
EP-0503537-A1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones THE UNIVERSITY OF VERMONT (US) 1992-09-16 EP claimed