SCHEMBL7827451

SCHEMBL7827451

CC(C)CNC(=O)Nc1snc(SCc2ccc(Cl)cc2)c1C(=O)O

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 15/20 0.62
HPGD P15428 2/20 0.40
HTT P42858 2/20 0.39
LMNA P02545 2/20 0.39
MEN1 O00255 2/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3087415 0.91 NTRK1 (0.76) NTRK1
SCHEMBL3087650 0.84 NTRK1 (0.74) NTRK1
SCHEMBL7833961 0.83 NTRK1 (0.48) NTRK1ALDH1A1
SCHEMBL3084738 0.82 NTRK1 (0.60) NTRK1
SCHEMBL3082246 0.82 NTRK1 (0.62) NTRK1HPGD
SCHEMBL3094633 0.81 NTRK1 (0.61) NTRK1KMT2A
SCHEMBL3096961 0.81 NTRK1 (0.61) NTRK1HPGD
SCHEMBL3087131 0.81 NTRK1 (0.72) NTRK1
SCHEMBL3085037 0.79 NTRK1 (0.59) NTRK1ALDH1A1
SCHEMBL3073533 0.79 NTRK1 (0.59) NTRK1HPGDLMNAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1084114-A1 ISOTHIAZOLE DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2001-03-21 EP disclosed
WO-1999062890-A1 ISOTHIAZOLE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 1999-12-09 WO disclosed