SCHEMBL7828089

SCHEMBL7828089

COc1ccc(S(C)(=O)=O)cc1C[C@H]1CCCN(N)[C@H]1c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 9/20 0.51
HTR6 P50406 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA7 P43166 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.38
DRD2 P14416 3/20 0.38
DRD3 P35462 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7833056 1.00 TACR1 (0.51) TACR1HTR6CA1CA2CA4
SCHEMBL7828087 1.00 TACR1 (0.51) TACR1HTR6CA1CA2CA4
SCHEMBL7817009 0.88 KMT2A (0.45) TACR1MEN1KMT2ADRD2DRD3
SCHEMBL7817012 0.88 KMT2A (0.45) TACR1MEN1KMT2ADRD2DRD3
SCHEMBL7051258 0.85 TACR1 (0.45) TACR1CA1CA2MEN1KMT2A
SCHEMBL27365754 0.83 TACR1 (0.53) TACR1MEN1KMT2A
SCHEMBL7817895 0.82 TACR1 (0.44) TACR1KMT2APOLBDRD2DRD3
Hydrochloric Acid SCHEMBL7837990 0.82 TACR1 (0.52) TACR1MEN1KMT2A
SCHEMBL9374751 0.82 TACR1 (0.49) TACR1
SCHEMBL9210577 0.82 TACR1 (0.49) TACR1MEN1KMT2APOLBDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655996-B1 SUBSTITUTED BENZYLAMINO NITROGEN CONTAINING NON-AROMATIC HETEROCYCLES PFIZER (US) 2001-11-07 EP claimed
EP-1114823-A2 Substituted benzylamino nitrogen containing non-aromatic heterocycles PFIZER INC. (US) 2001-07-11 EP claimed