SCHEMBL7828569

SCHEMBL7828569

[CH]=CC(=O)c1ccccc1OC

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.62
MAOB P27338 2/20 0.54
CTSD P07339 1/20 0.53
GPR52 Q9Y2T5 1/20 0.53
ABCB1 P08183 1/20 0.53
STAT3 P40763 1/20 0.50
AR P10275 2/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
NPC1 O15118 3/20 0.49
HTT P42858 2/20 0.49
RAB9A P51151 1/20 0.49
KCNK3 O14649 1/20 0.47
KCNK9 Q9NPC2 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31167606 0.84 ABCG2 (0.77) ABCG2MAOBCTSDGPR52ABCB1
SCHEMBL31561740 0.82 ABCG2 (0.64) ABCG2MAOBCTSDGPR52ABCB1
SCHEMBL1697561 0.82 ABCG2 (0.64) ABCG2MAOBCTSDGPR52ABCB1
SCHEMBL29954715 0.82 ABCG2 (0.64) ABCG2MAOBCTSDGPR52ABCB1
SCHEMBL9178467 0.82 ABCG2 (0.64) ABCG2MAOBCTSDGPR52ABCB1
SCHEMBL7469828 0.82 ABCG2 (0.64) ABCG2MAOBCTSDGPR52ABCB1
SCHEMBL15821571 0.81 ABCG2 (0.62) ABCG2MAOBCTSDGPR52ABCB1
Water SCHEMBL3048073 0.81 ABCG2 (0.62) ABCG2MAOBCTSDGPR52ABCB1
SCHEMBL15563363 0.80 CA12 (0.69) ABCG2MAOBCTSDGPR52ABCB1
SCHEMBL15563364 0.80 CA12 (0.69) ABCG2MAOBCTSDGPR52ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686636-B1 TRICYCLIC BENZAZEPINE AND BENZOTHIAZEPINE DERIVATIVES MEIJI SEIKA CO (JP) 2001-04-04 EP disclosed
US-5840895-A INTERMEDIATES FOR ANTIALLERGENS MEIJI SEIKA KABUSHIKI KAISHA (JP) 1998-11-24 US disclosed
US-5686442-A ANTIALLERGENS MEIJI SEIKA KABUSHIKI KAISHA (JP) 1997-11-11 US disclosed
EP-0686636-A1 TRICYCLIC BENZAZEPINE AND BENZOTHIAZEPINE DERIVATIVES MEIJI SEIKA KABUSHIKI KAISHA (JP) 1995-12-13 EP disclosed