SCHEMBL7828579

SCHEMBL7828579

Cc1cccc2c(C[O])cccc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.59
CYP2A6 P11509 3/20 0.59
ALDH1A1 P00352 2/20 0.44
CYP3A4 P08684 2/20 0.36
CYP2C19 P33261 2/20 0.36
DAO P14920 1/20 0.36
CYP2D6 P10635 1/20 0.36
TAAR1 Q96RJ0 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
AR P10275 1/20 0.35
GABRA1 P14867 2/20 0.34
GABRB2 P47870 2/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
HTR2A P28223 1/20 0.34
CES1 P23141 2/20 0.34
TYMP P19971 1/20 0.34
CES2 O00748 1/20 0.34
KDM1A O60341 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3090285 0.86 CYP1A2 (0.59) CYP1A2CYP2A6ALDH1A1CYP3A4CYP2C19
SCHEMBL599157 0.84 CYP1A2 (0.62) CYP1A2CYP2A6ALDH1A1DAOTAAR1
SCHEMBL14496815 0.82 CYP1A2 (0.59) CYP1A2CYP2A6ALDH1A1CYP3A4CYP2C19
SCHEMBL10900222 0.77 CYP1A2 (0.59) CYP1A2CYP2A6ALDH1A1CYP3A4CYP2C19
SCHEMBL15345377 0.77 CYP1A2 (0.59) CYP1A2CYP2A6ALDH1A1CYP3A4CYP2C19
SCHEMBL424167 0.77 CYP1A2 (1.00) CYP1A2CYP2A6ALDH1A1CYP3A4HPGD
SCHEMBL29463284 0.77 CYP1A2 (1.00) CYP1A2CYP2A6ALDH1A1CYP3A4HPGD
SCHEMBL395673 0.76 ESR1 (0.44) CYP1A2CYP2A6ALDH1A1TAAR1HSD17B10
SCHEMBL392411 0.75
SCHEMBL5235003 0.75 CYP1A2 (0.50) CYP1A2CYP2A6ALDH1A1HPGDPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0454501-B1 Benzylidenethiazolidine derivatives, their preparation and their use for the inhibition of lipid peroxides SANKYO CO (JP) 2001-09-05 EP disclosed
EP-0839812-A1 Preparation of benzylthiazolidine derivatives Sankyo Company Limited (JP) 1998-05-06 EP disclosed
US-5387596-A Treating arteriosclerosis SANKYO COMPANY, LIMITED (JP) 1995-02-07 US disclosed
EP-0454501-A2 Benzylidenethiazolidine derivatives, their preparation and their use for the inhibition of lipid peroxides Sankyo Company Limited (JP) 1991-10-30 EP disclosed