SCHEMBL7828679

SCHEMBL7828679

CN1C(=O)CCc2cc(OC(F)F)c(CNC3CCCN(C(=O)OC(C)(C)C)C3c3ccccc3)cc21

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 1/20 0.39
TACR1 P25103 9/20 0.38
TRPV1 Q8NER1 6/20 0.36
KDM1A O60341 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TMEM97 Q5BJF2 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6604442 1.00 HCRTR2 (0.39) HCRTR2TACR1TRPV1KDM1AMEN1
SCHEMBL8596137 0.94 HCRTR2 (0.39) HCRTR2TACR1TRPV1KDM1AMEN1
SCHEMBL6607716 0.94 HCRTR2 (0.39) HCRTR2TACR1TRPV1KDM1AMEN1
SCHEMBL6605255 0.89 HCRTR2 (0.39) HCRTR2TACR1TRPV1KDM1AMEN1
SCHEMBL8664244 0.88 TACR1 (0.45) HCRTR2TACR1TRPV1KDM1A
SCHEMBL6606866 0.88 TACR1 (0.45) HCRTR2TACR1TRPV1KDM1A
SCHEMBL7030644 0.88 TACR1 (0.44) HCRTR2TACR1KDM1AMEN1KMT2A
SCHEMBL6606522 0.88 TACR1 (0.44) HCRTR2TACR1KDM1AMEN1KMT2A
SCHEMBL7033824 0.86 TACR1 (0.43) HCRTR2TACR1KDM1A
SCHEMBL6603700 0.86 TACR1 (0.43) HCRTR2TACR1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840732-B1 SUBSTITUTED BENZOLACTAM COMPOUNDS AS SUBSTANCE P ANTAGONISTS PFIZER (US) 2001-03-07 EP disclosed