SCHEMBL7833859

SCHEMBL7833859

O=C1NC(=O)C(Cc2ccc(OCc3cn4ccccc4n3)cc2)S1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.56
PPARG P37231 8/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
FFAR1 O14842 11/20 0.54
PPARA Q07869 6/20 0.54
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7833990 0.91 PPARG (0.57) PPARGFFAR1PPARA
SCHEMBL7822745 0.78 KDM4E (0.53) KDM4ESMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL8314978 0.77 FFAR1 (0.70) PPARGFFAR1PPARAALDH1A1
SCHEMBL1299855 0.77 FFAR1 (0.80) PPARGFFAR1PPARAALDH1A1
SCHEMBL8312136 0.76 FFAR1 (0.87) PPARGFFAR1PPARAALDH1A1
SCHEMBL7454600 0.76 FFAR1 (0.62) PPARGFFAR1PPARA
SCHEMBL10365333 0.74 FFAR1 (0.63) PPARGFFAR1PPARAALDH1A1
SCHEMBL1072226 0.74 FFAR1 (0.77) PPARGFFAR1PPARAALDH1A1
SCHEMBL9570853 0.74 FFAR1 (0.69) PPARGFFAR1PPARAALDH1A1
SCHEMBL8957444 0.74 FFAR1 (0.69) PPARGFFAR1PPARAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676398-B1 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO CO (JP) 2001-10-24 EP disclosed
US-6117893-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 2000-09-12 US disclosed
EP-1022274-A1 Oxazolidinedione and Thiazolidinedione derivatves, their preparation and their use Sankyo Company Limited (JP) 2000-07-26 EP disclosed
US-5977365-A HYPOGLYCEMIC AGENTS SANKYO COMPANY, LIMITED (JP) 1999-11-02 US disclosed
US-5962470-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 1999-10-05 US disclosed
US-5834501-A TREATING DIABETES OR HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 1998-11-10 US disclosed
US-5739345-A HYPOGLYCEMIC AND ANTIDIABETIC AGENTS SANKYO COMPANY, LIMITED (JP) 1998-04-14 US disclosed
US-5624935-A ANTIDIABETIC AGENTS, HYPOGLYCEMIC AGENTS OR ANTILIPEMIC AGENTS SANKYO COMPANY, LIMITED 1997-04-29 US disclosed
EP-0676398-A2 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO COMPANY LIMITED (JP) 1995-10-11 EP disclosed