SCHEMBL7834787

SCHEMBL7834787

Oc1c(C(=S)NCc2ccc(Cl)cc2)cnc2ccc(CN3CCOCC3)cc12

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MELK Q14680 3/20 0.46
KCNH2 Q12809 5/20 0.44
LMNA P02545 2/20 0.44
POLA1 P09884 2/20 0.44
ALDH1A1 P00352 2/20 0.41
F10 P00742 1/20 0.41
KDM4E B2RXH2 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PDE1B Q01064 1/20 0.41
EGFR P00533 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201283 0.89 KCNH2 (0.54) MELKKCNH2POLA1ALDH1A1F10
SCHEMBL6665763 0.85 KCNH2 (0.54) MELKKCNH2POLA1ALDH1A1F10
SCHEMBL7843275 0.82 QPCT (0.39) ALDH1A1EGFR
SCHEMBL6667972 0.79 TRPV1 (0.40) ALDH1A1EGFR
SCHEMBL6669690 0.78 KCNH2 (0.50) KCNH2POLA1ALDH1A1F10NPC1
SCHEMBL6713757 0.77 EGLN1 (0.51) KCNH2POLA1ALDH1A1PDE1BNPC1
SCHEMBL6670929 0.76 POLA1 (0.50) KCNH2POLA1ALDH1A1NPC1RAB9A
SCHEMBL6339478 0.75 KCNH2 (0.51) KCNH2LMNAPOLA1F10
SCHEMBL6200011 0.75 KCNH2 (0.53) KCNH2POLA1ALDH1A1F10
SCHEMBL6770778 0.75 KCNH2 (0.53) KCNH2POLA1ALDH1A1F10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140850-A1 QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2001-10-10 EP disclosed
US-6248739-B1 DNA POLYMERASE INHIBITORS EFFECTIVE AGAINST HERPESVIRUSES PHARMACIA & UPJOHN COMPANY 2001-06-19 US disclosed
WO-2000040561-A1 QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2000-07-13 WO disclosed