SCHEMBL7834814

SCHEMBL7834814

OCc1nc2cc(-c3ncc[nH]3)ccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.46
NPSR1 Q6W5P4 1/20 0.42
NISCH Q9Y2I1 2/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MTOR P42345 1/20 0.39
ADK P55263 1/20 0.39
PARP1 P09874 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP19A1 P11511 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
RHEB Q15382 1/20 0.37
TLR9 Q9NR96 1/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
MAPK14 Q16539 1/20 0.35
SMPD3 Q9NY59 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL548479 0.89 NISCH (0.42) NISCHKDM4EALDH1A1MTORADK
SCHEMBL548422 0.89 NISCH (0.42) NISCHKDM4EALDH1A1MTORADK
SCHEMBL548266 0.86 POLB (0.50) TDP1NISCHKDM4ECYP1A2CYP3A4
SCHEMBL548416 0.86 POLB (0.46) TDP1NISCHKDM4EALDH1A1MTOR
SCHEMBL549255 0.85 NISCH (0.40) NISCHKDM4EALDH1A1MTORADK
SCHEMBL549254 0.85 NISCH (0.40) NISCHKDM4EALDH1A1MTORADK
SCHEMBL5304913 0.85 POLB (0.49) TDP1NISCHKDM4ECYP1A2CYP3A4
SCHEMBL548311 0.83 CYP1A2 (0.39) NISCHKDM4EALDH1A1MTORADK
SCHEMBL548310 0.83 CYP1A2 (0.39) NISCHKDM4EALDH1A1MTORADK
SCHEMBL5311172 0.81 CYP1A2 (0.48) TDP1NISCHKDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894795-B1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-06 EP disclosed
EP-0894795-A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-02-03 EP disclosed