SCHEMBL7839255

SCHEMBL7839255

COc1ccc(-c2ccc(Cl)cc2)c(COc2ccc(I)cc2)c1.Oc1ccc(I)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.48
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
APP P05067 5/20 0.47
MAPT P10636 3/20 0.46
ALOX12 P18054 2/20 0.46
ALOX15 P16050 1/20 0.46
FFAR1 O14842 3/20 0.46
FFAR4 Q5NUL3 3/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
KDM4E B2RXH2 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CNR1 P21554 1/20 0.42
CYP2C19 P33261 1/20 0.42
CNR2 P34972 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5516525 0.95 APP (0.51) NPSR1MEN1KMT2AAPPMAPT
SCHEMBL7840330 0.83 MAPT (0.42) NPSR1MEN1KMT2AAPPMAPT
SCHEMBL10293539 0.83 FFAR1 (0.59) NPSR1MEN1KMT2AMAPTALOX12
SCHEMBL13165361 0.81 FFAR1 (0.46) NPSR1MEN1KMT2AMAPTALOX12
SCHEMBL791494 0.79 MEN1 (0.50) NPSR1MEN1KMT2AMAPTALOX12
SCHEMBL10138010 0.77 CYP11B1 (0.47) MEN1KMT2AAPPMAPTKDM4E
SCHEMBL5521150 0.77 MEN1 (0.51) NPSR1MEN1KMT2AMAPTALOX12
SCHEMBL6700683 0.76 MAPT (0.46) NPSR1MEN1KMT2AMAPTALOX12
SCHEMBL27553691 0.75 FFAR1 (0.43) NPSR1MEN1KMT2AMAPTALOX12
SCHEMBL5510993 0.74 MEN1 (0.48) NPSR1MEN1KMT2AMAPTALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1162196-A1 FUSED-RING COMPOUNDS AND USE THEREOF AS DRUGS JAPAN TOBACCO INC. (JP) 2001-12-12 EP disclosed