SCHEMBL7841422

SCHEMBL7841422

O=C(NCc1ccc(Cl)cc1)c1cnc2ccc(CC3CCOCC3)cc2c1O

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.45
RXFP1 Q9HBX9 1/20 0.44
CNR2 P34972 11/20 0.41
CYP2C9 P11712 6/20 0.41
CYP1A2 P05177 4/20 0.41
CYP3A4 P08684 4/20 0.41
EGLN1 Q9GZT9 1/20 0.41
CYP2C19 P33261 5/20 0.41
CYP2D6 P10635 4/20 0.41
TP53 P04637 1/20 0.41
NR3C1 P04150 1/20 0.40
CNR1 P21554 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6766761 0.86 MAPK1 (0.45) MAPK1RXFP1CNR2CYP2C9CYP1A2
SCHEMBL6716698 0.84 EGLN1 (0.47) MAPK1RXFP1EGLN1
SCHEMBL6670932 0.84 MAPK1 (0.41) MAPK1EGLN1
SCHEMBL6713866 0.83 EGLN1 (0.46) MAPK1RXFP1CNR2CYP2C9CYP1A2
SCHEMBL6201283 0.83 KCNH2 (0.54) RXFP1
SCHEMBL6198849 0.82 EGLN1 (0.51) RXFP1CNR2CYP2C9CYP1A2CYP3A4
SCHEMBL6699267 0.82 MAPK1 (0.42) MAPK1RXFP1CNR2CYP2C9CYP1A2
SCHEMBL6200824 0.82 EGLN1 (0.48) CYP2C9CYP1A2CYP3A4EGLN1CYP2C19
SCHEMBL6669425 0.81 MAPK1 (0.45) MAPK1RXFP1EGLN1
SCHEMBL6194761 0.81 POLA1 (0.54) CNR2CYP2C9CYP1A2CYP3A4EGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140850-A1 QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2001-10-10 EP disclosed
US-6248739-B1 DNA POLYMERASE INHIBITORS EFFECTIVE AGAINST HERPESVIRUSES PHARMACIA & UPJOHN COMPANY 2001-06-19 US disclosed
WO-2000040561-A1 QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2000-07-13 WO disclosed