SCHEMBL7844102

SCHEMBL7844102

COC(=O)CN1CCCC(Nc2cc(Nc3cccc(Br)c3)ncn2)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.48
ERBB3 P21860 1/20 0.48
TNNI3K Q59H18 1/20 0.42
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41
TUBB4B P68371 1/20 0.41
TUBB3 Q13509 1/20 0.41
TUBB2A Q13885 1/20 0.41
TUBB8 Q3ZCM7 1/20 0.41
TUBA3E Q6PEY2 1/20 0.41
TUBA1A Q71U36 1/20 0.41
TUBA1C Q9BQE3 1/20 0.41
TUBB6 Q9BUF5 1/20 0.41
TUBB2B Q9BVA1 1/20 0.41
TUBB1 Q9H4B7 1/20 0.41
ERBB2 P04626 4/20 0.40
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7853903 0.93 EGFR (0.48) EGFRERBB3TNNI3KTUBB4ATUBB
SCHEMBL7851124 0.90 EGFR (0.44) EGFRERBB3TNNI3KTUBB4ATUBB
SCHEMBL7854732 0.89 EGFR (0.47) EGFRERBB3TNNI3KTUBB4ATUBB
SCHEMBL7696986 0.89 EGFR (0.51) EGFRERBB3TNNI3KTUBB4ATUBB
SCHEMBL7855967 0.87 EGFR (0.43) EGFRERBB3TUBB4ATUBBTUBA3C
SCHEMBL7851215 0.83 EGFR (0.44) EGFRTNNI3KTUBB4ATUBBTUBA3C
SCHEMBL7850948 0.82 EGFR (0.47) EGFRERBB3TNNI3KTUBB4ATUBB
SCHEMBL7851577 0.82 EGFR (0.52) EGFRERBB3TNNI3KTUBB4ATUBB
SCHEMBL7581148 0.81 EGFR (0.53) EGFRERBB2
SCHEMBL7855902 0.80 EGFR (0.46) EGFRERBB3TUBB4ATUBBTUBA3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163242-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM Boehringer Ingelheim Pharma KG (DE) 2001-12-19 EP disclosed
WO-2000055162-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-21 WO disclosed