SCHEMBL7845256

SCHEMBL7845256

CC[SiH](CC)CC.CN1CCC(c2c[nH]c3ccc([N+](=O)[O-])cc23)CC1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 14/20 0.55
HTR1B P28222 14/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
THPO P40225 1/20 0.55
HTR1A P08908 4/20 0.51
HTR1F P30939 3/20 0.51
APP P05067 1/20 0.50
MAPT P10636 1/20 0.50
BLM P54132 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
SLC6A4 P31645 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6640192 0.92 HTR1D (0.63) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL3337136 0.83 APP (0.57) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL8820381 0.80 HTR1D (0.47) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL9836165 0.79 KDM4E (0.63) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL17060365 0.79 HSP90AA1 (0.54) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL15712312 0.78 HSP90AA1 (0.56) MAPTSLC6A4
SCHEMBL5369303 0.77 HTR1D (0.50) HTR1DHTR1BCYP1A2CYP3A4CYP2D6
SCHEMBL9836911 0.77 HTR2C (0.55) APPSLC6A4
SCHEMBL7489905 0.76 HTR1D (0.76) HTR1DHTR1BHTR1AHTR1F
Phosphoric Acid SCHEMBL7867279 0.76 CYP1A2 (0.46) HTR1DHTR1BCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089993-A1 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2001-04-11 EP disclosed
WO-2000000487-A1 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2000-01-06 WO disclosed