SCHEMBL7846052

SCHEMBL7846052

NCCN(Cc1ccc(CN(Cc2ccccn2)C2CCCc3cccnc32)cc1)S(=O)(=O)c1ccccc1[N+](=O)[O-]

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 20/20 0.56
CYP2D6 P10635 3/20 0.43
CYP3A4 P08684 2/20 0.43
CHRM2 P08172 1/20 0.43
DRD2 P14416 1/20 0.43
OPRM1 P35372 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3314059 0.94 CXCR4 (0.56) CXCR4CYP2D6CYP3A4CHRM2DRD2
Trifluoroacetic Acid SCHEMBL4541649 0.88 CXCR4 (0.49) CXCR4CYP2D6CYP3A4KCNH2
SCHEMBL4074278 0.84 CXCR4 (0.52) CXCR4CYP2D6CYP3A4CHRM2DRD2
SCHEMBL4250911 0.83 CXCR4 (0.47) CXCR4CYP2D6CYP3A4CHRM2DRD2
SCHEMBL3312985 0.82 CXCR4 (0.48) CXCR4CYP2D6CYP3A4
SCHEMBL3312846 0.81 HDAC6 (0.48) CXCR4CYP2D6CYP3A4
SCHEMBL3314317 0.79 HDAC6 (0.46) CXCR4CYP2D6CYP3A4
SCHEMBL30338222 0.78 CXCR4 (0.70) CXCR4CYP2D6CYP3A4
SCHEMBL28610931 0.78 CXCR4 (0.70) CXCR4CYP2D6CYP3A4
SCHEMBL3313097 0.76 HDAC6 (0.42) CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163238-A1 CHEMOKINE RECPETOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC. (CA) 2001-12-19 EP disclosed
WO-2000056729-A1 CHEMOKINE RECPETOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC. (CA) 2000-09-28 WO disclosed