SCHEMBL7846955

SCHEMBL7846955

Nc1nc2[nH]cc(CCCc3ccc(C(=O)O)cc3)c2c(=O)[nH]1

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TYMS P04818 18/20 0.66
DHFR P00374 2/20 0.60
FOLR1 P15328 2/20 0.60
SLC19A1 P41440 2/20 0.60
SLC46A1 Q96NT5 2/20 0.60
FOLR2 P14207 1/20 0.60
GART P22102 1/20 0.60
ATIC P31939 1/20 0.60
SHMT1 P34896 1/20 0.60
FRK P42685 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2260428 0.93 TYMS (0.69) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL2260030 0.92 TYMS (0.67) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL17518729 0.85 TYMS (0.62) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL18551642 0.84 TYMS (0.64) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL13659935 0.83 TYMS (0.63) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL7836050 0.82 GART (0.90) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL20780521 0.82 TYMS (0.56) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL2260032 0.82 TYMS (0.68) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL28417050 0.82 TYMS (0.45) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL7836419 0.81 NAMPT (0.56) TYMSDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112442038-B Industrial preparation method of pemetrexed disodium 德州德药制药有限公司 2022-09-02 CN claimed
CN-112174970-B Method for preparing pemetrexed disodium with high yield 德州德药制药有限公司 2022-06-07 CN claimed
CN-112442038-A Industrial preparation method of pemetrexed disodium 德州德药制药有限公司 2021-03-05 CN claimed
CN-112174970-A Method for preparing pemetrexed disodium in high yield 德州德药制药有限公司 2021-01-05 CN claimed
CN-112442038-B Industrial preparation method of pemetrexed disodium 德州德药制药有限公司 2022-09-02 CN disclosed
CN-112174970-B Method for preparing pemetrexed disodium with high yield 德州德药制药有限公司 2022-06-07 CN disclosed
CN-112442038-A Industrial preparation method of pemetrexed disodium 德州德药制药有限公司 2021-03-05 CN disclosed
CN-112174970-A Method for preparing pemetrexed disodium in high yield 德州德药制药有限公司 2021-01-05 CN disclosed
EP-1105396-A1 PROCESS FOR THE PREPARATION OF PYRROLO[2,3-D]PYRIMIDINES The Trustees of Princeton University (US) 2001-06-13 EP disclosed
US-6066732-A Process for the preparation of pyrrolo[2,3-d]pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2000-05-23 US disclosed
WO-2000011004-A1 PROCESS FOR THE PREPARATION OF PYRROLO[2,3-D]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2000-03-02 WO disclosed