SCHEMBL7848504

SCHEMBL7848504

Cc1ccc(Nc2cc(N3CCOCC3)cc(C(F)(F)F)c2)cc1NC(=O)c1ccc(Cl)nc1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 6/20 0.64
ALDH1A1 P00352 1/20 0.60
GAA P10253 1/20 0.60
MAPT P10636 1/20 0.57
BRAF P15056 10/20 0.55
MAPK14 Q16539 1/20 0.55
LYN P07948 2/20 0.53
KIT P10721 1/20 0.53
TDP1 Q9NUW8 1/20 0.51
RAF1 P04049 1/20 0.50
KDM4E B2RXH2 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5897191 0.91 CSF1R (0.74) CSF1RALDH1A1GAAMAPTBRAF
SCHEMBL7850678 0.89 MAPT (0.60) CSF1RALDH1A1GAAMAPTMAPK14
SCHEMBL5897317 0.82 MAPK14 (0.66) CSF1RMAPTBRAFMAPK14TDP1
SCHEMBL2975514 0.79 MAPT (0.64) CSF1RALDH1A1GAAMAPTBRAF
SCHEMBL4878747 0.78 CSF1R (0.52) CSF1RALDH1A1MAPTBRAFMAPK14
SCHEMBL7827478 0.78 CSF1R (0.52) CSF1RMAPTBRAFMAPK14LYN
SCHEMBL7851337 0.77 MAPK14 (0.52) MAPTBRAFMAPK14
SCHEMBL5897092 0.76 MAPK14 (0.71) MAPTBRAFMAPK14TDP1RAF1
SCHEMBL7822467 0.76 BRAF (0.54) CSF1RBRAFMAPK14LYNKIT
SCHEMBL25238622 0.76 CSF1R (1.00) CSF1RBRAFMAPK14LYNKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102750-A1 AMIDE DERIVATIVES USEFUL AS INHIBITORS OF THE PRODUCTION OF CYTOKINES AstraZeneca AB (SE) 2001-05-30 EP disclosed
WO-2000007991-A1 AMIDE DERIVATIVES USEFUL AS INHIBITORS OF THE PRODUCTION OF CYTOKINES ASTRAZENECA AB (SE) 2000-02-17 WO disclosed