SCHEMBL7850671

SCHEMBL7850671

CN(C)c1ccc(CN2CCC(CCOc3ccc4c(c3)CN(Cc3ccccc3)CCC4)CC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.54
MCHR1 Q99705 1/20 0.51
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
ACACB O00763 2/20 0.47
ACHE P22303 5/20 0.45
MAOA P21397 3/20 0.44
BCHE P06276 2/20 0.44
MAOB P27338 2/20 0.44
BACE1 P56817 1/20 0.44
SIGMAR1 Q99720 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7848542 0.99 HRH3 (0.53) HRH3MCHR1DRD2DRD4ACACB
SCHEMBL7838701 0.92 HRH3 (0.62) HRH3MCHR1DRD2DRD4ACACB
SCHEMBL7847862 0.88 HRH3 (0.52) HRH3MCHR1DRD2DRD4ACACB
Hydrochloric Acid SCHEMBL7849060 0.87 HRH3 (0.52) HRH3MCHR1DRD2DRD4ACACB
SCHEMBL7846368 0.86 HRH3 (0.54) HRH3MCHR1DRD2DRD4ACACB
Diethylamine SCHEMBL7847864 0.85 HRH3 (0.52) HRH3MCHR1DRD2DRD4ACACB
Diethylamine SCHEMBL7849064 0.84 HRH3 (0.51) HRH3MCHR1DRD2DRD4ACACB
Hydrochloric Acid SCHEMBL7846814 0.83 HRH3 (0.48) HRH3MCHR1DRD2DRD4ACACB
SCHEMBL7838474 0.83 HRH3 (0.59) HRH3MCHR1DRD2DRD4ACACB
Hydrochloric Acid SCHEMBL7846320 0.83 HRH3 (0.57) HRH3MCHR1ACHEMAOABCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1122252-A1 NITROGENOUS FUSED HETEROCYCLE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-08 EP claimed
EP-1122252-A1 NITROGENOUS FUSED HETEROCYCLE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-08 EP disclosed