SCHEMBL7853019

SCHEMBL7853019

O=C(NC1CCCC1)C(OC(=O)C(F)(F)F)C1CCCN1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
EPHX1 P07099 1/20 0.33
SLC6A3 Q01959 3/20 0.32
TSHR P16473 2/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
DHFR P00374 1/20 0.32
EPHX2 P34913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7851340 0.99 MEN1 (0.36) MEN1KMT2APDK1PDK2PDK3
Trifluoroacetic Acid SCHEMBL7853017 0.76 DPP4 (0.35) PDK1PDK2PDK3PDK4EPHX1
Trifluoroacetic Acid SCHEMBL7851338 0.75 EPHX1 (0.36) PDK1PDK2PDK3PDK4EPHX1
SCHEMBL9046184 0.71 EPHX1 (0.43) EPHX1EPHX2
SCHEMBL7851143 0.71 EPHX1 (0.43) EPHX1EPHX2
Hydrochloric Acid SCHEMBL7853040 0.70 EPHX1 (0.42) EPHX1SLC6A3TSHRSLC6A2EPHX2
Hydrochloric Acid SCHEMBL7845299 0.70 EPHX1 (0.42) EPHX1SLC6A3TSHRSLC6A2EPHX2
Hydrochloric Acid SCHEMBL7853365 0.70 EPHX1 (0.42) EPHX1SLC6A3TSHRSLC6A2EPHX2
SCHEMBL4328004 0.68
SCHEMBL9047402 0.67 KMT2A (0.36) KMT2AEPHX1SLC6A3TSHRSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709373-B1 PYRROLIDINE DERIVATIVE ZAIDAN HOJIN BISEIBUTSU (JP) 2001-10-17 EP disclosed
US-5965556-A KETO-ACID AMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND METHODS FOR INHIBITING THE ACTIVITY OF SERINE PROTEASE OR THIOL PROTEASE BY ADMINISTERING THE DERIVATIVE TO A MAMMAL; ALZHEIMER'S DISEASE ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYUKAI (JP) 1999-10-12 US disclosed
US-5756763-A ENZYME INHIBITOR ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYUKAI (JP) 1998-05-26 US disclosed
EP-0709373-A1 NOVEL PYRROLIDINE DERIVATIVE ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1996-05-01 EP disclosed