SCHEMBL7860009

SCHEMBL7860009

C=C(c1cc2cc(S(C)(=O)=O)ccc2n1CC)N1CCOc2ccc(-c3ccc4nc(C)[nH]c4c3)cc2C1

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 16/20 0.51
PRKDC P78527 1/20 0.36
CREBBP Q92793 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3756772 0.92 PIK3CA (0.57) PIK3CAPRKDCCREBBP
SCHEMBL3762451 0.84 PIK3CA (0.60) PIK3CAPRKDCCREBBP
SCHEMBL3754736 0.81 PIK3CA (0.61) PIK3CAPRKDC
SCHEMBL3748041 0.79 PIK3CA (0.62) PIK3CAPRKDCCREBBP
SCHEMBL3755298 0.79 PIK3CA (0.76) PIK3CA
SCHEMBL3757004 0.78 PIK3CA (0.65) PIK3CAPRKDCCREBBP
Hydrochloric Acid SCHEMBL3762167 0.77 PIK3CA (0.64) PIK3CAPRKDCCREBBP
SCHEMBL3753793 0.77 PIK3CA (0.76) PIK3CA
SCHEMBL3755378 0.77 PIK3CA (0.77) PIK3CAPRKDCCREBBP
SCHEMBL3755685 0.77 PIK3CA (0.64) PIK3CAPRKDCCREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118208-A1 BENZOXAZEPIN-4- (5H) -YL DERIVATIVES AND THEIR USE TO TREAT CANCER EXELIXIS, INC. (US) 2010-10-14 WO disclosed